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3-{1-[5-(naphthalen-1-yl)-1,2,4-triazin-3-yl]piperidin-3-yl}propan-1-ol
1-[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
[(2-cyclohexylpyrimidin-5-yl)methyl](1H-imidazol-2-ylmethyl)methylamine
N-{3-[(2-ethylphenyl)carbamoyl]phenyl}-1-methyl-1H-pyrrole-2-carboxamide
(2R)-2-hydroxy-1-{4-[(2-hydroxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-phenylethan-1-one
2-amino-6-(2-hydroxypropan-2-yl)-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]pyridine-3-carbonitrile
4-[(2S)-1-(3,5-dichloro-4-methylbenzoyl)pyrrolidine-2-carbonyl]morpholine
4-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1,4-diazepane-1-carboxamide
[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl](pyridin-2-yl)methanol
N-(1-methoxybutan-2-yl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
5-benzyl-4-(3-hydroxypropanoyl)-1-(2-phenylphenyl)piperazin-2-one
N-{3-[({1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}carbamoyl)amino]phenyl}acetamide
{[(1R,5S,6S)-3-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
2-[3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)phenyl]-4-methyl-1,2-dihydrophthalazin-1-one
N-[(3S,4R)-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-(ethylsulfanyl)-5-({8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)pyrimidine
5-ethyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-oxazole-4-carboxamide
N-(furan-3-ylmethyl)-5-{1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-N,2,2,6,6-pentamethylpiperidin-4-amine
N-{1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-(2-chlorophenyl)ethyl}-N-methylfuran-2-carboxamide
1-(furan-2-yl)-2-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]ethane-1,2-dione
4-[(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)methyl]pyridine
[(2,3-difluoro-4-methylphenyl)methyl](methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-2,3-dimethoxy-N-(pyridin-3-ylmethyl)benzamide
2-[(1S,5R)-3-(2,3-dihydro-1H-indene-5-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-(1-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
2-methyl-4-(4-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}phenyl)butan-2-ol
7-(2-cyclohexylethyl)-2-(4-methyl-1,3-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrimidin-2-amine
2-(carbamoylamino)-3-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]butanamide
4-{[5-(2-methyl-1,3-thiazol-4-yl)thiophen-2-yl]sulfonyl}piperazine-2-carboxylic acid
2-(4-{6-[(propan-2-yl)amino]pyrimidin-4-yl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
N,N-bis(2-ethoxyethyl)-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
N-methyl-N-{2-phenyl-1-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]ethyl}oxane-4-carboxamide
N4-[1-(3,4-dimethoxyphenyl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
5-({1-[(4-ethylphenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(1-benzyl-1H-pyrazol-3-yl)-2-{4-[4-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
3-{imidazo[1,2-a]pyridin-2-yl}-1-(thiomorpholin-4-yl)propan-1-one
1-{5-[(4-hydroxyphenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
3-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}pyridine
2-methyl-8-[(3-methylthiophen-2-yl)sulfonyl]-2,8-diazaspiro[4.5]decane
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-[(2R)-pyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4aS,8aR)-1-(carboxymethyl)-6-[(3-methylphenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
5-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}-1-(3-phenylpropyl)piperidin-2-one
N-(4-chloro-1-methyl-1H-indazol-3-yl)-2-[4-(5-methoxypyridin-3-yl)-1H-pyrazol-1-yl]acetamide
4-[2-(dimethylamino)acetamido]-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}benzamide
[(1-ethyl-1H-imidazol-2-yl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amine
2-{[(5-tert-butyl-2-methoxyphenyl)carbamoyl]amino}acetamide
4-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-yl]-5-(2-methylphenyl)-2-(pyridin-4-yl)pyrimidine