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2-{2-[(1H-indol-2-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
13-(1H-indol-4-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
(3R,4R)-4-{[2-(1H-indol-3-yl)ethyl]amino}-1-(4-methoxybenzoyl)pyrrolidin-3-ol
N-[1-({[(1-benzyl-1H-pyrazol-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
3-{[(furan-2-ylmethyl)(prop-2-en-1-yl)amino]methyl}-5-methyl-1H-indole-2-carboxylic acid
3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-[4-(morpholine-4-carbonyl)phenyl]urea
5-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2-carbonitrile
N-cyclopropyl-5-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-[2-(3-fluorophenoxy)acetyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
[(4-{1-[(3-chloropyridin-4-yl)methyl]pyrrolidin-2-yl}phenyl)methyl]dimethylamine
(3S,4S)-1-[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
[(4,5-dimethylfuran-2-yl)methyl]({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-(morpholin-3-yl)acetamide
2-[4-(4-fluorophenoxy)piperidine-1-carbonyl]-1-methyl-1H-indole
N-(pyridin-2-ylmethyl)-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidine-4-carboxamide
2-{[(4aS,8aR)-1-(3-methoxypropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]methyl}benzonitrile
9-[1-(4-fluorophenyl)cyclopropanecarbonyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(cyclobutylmethyl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3-(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
ethyl 1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-2-carboxylate
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-6-(methoxymethyl)pyrimidin-4-amine
3-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-1H-pyrazol-5-amine
4-[(1R)-1-(4-fluorophenyl)ethyl]-3-(1-methylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[2-(N-methylmethanesulfonamido)ethyl]urea
7-chloro-2-(furan-2-yl)-8-methyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]quinoline-4-carboxamide
methyl 1-{[(1-methyl-1H-1,2,3-triazol-4-yl)carbamoyl]methyl}-1H-indazole-3-carboxylate
N-{4-[2-(2-chlorophenyl)-1H-imidazol-1-yl]phenyl}acetamide
N-[1-(4-methylphenyl)ethyl]-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-yl}acetamide
2-methyl-4-(3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}phenyl)butan-2-ol
8-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1-oxa-8-azaspiro[4.5]decane
(3aR,6aR)-2-cyclobutanecarbonyl-5-(5-ethyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
1-{[1-(1-hexylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}azetidin-3-ol
2-(2-chlorophenyl)-2-hydroxy-1-{4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}ethan-1-one
3-[3-(dimethylamino)propyl]-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(1H-imidazol-2-yl)benzoyl]-3-phenylpiperazine
ethyl 3-({2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}amino)propanoate
1-methyl-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-N-(pyridin-4-ylmethyl)piperidin-4-amine
2-chloro-4-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
3-{[(dicyclopropylmethyl)(methyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N,8-dimethyl-N-(2-phenylethyl)-3-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}imidazo[1,2-a]pyridine-2-carboxamide
2-[(3-chlorophenyl)methyl]-N-[3-(morpholin-4-yl)propyl]-1,3-benzoxazole-6-carboxamide
N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
N-{2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxoethyl}methanesulfonamide
7-(1,3-benzothiazol-2-yl)-N-ethyl-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylfuran-3-carboxamide
2-{[(2R,5S)-2,5-dimethylpyrrolidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-({[2-(4-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]benzamide