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4-chloro-N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-1-methyl-1H-pyrazole-5-carboxamide
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-5-[(pyridin-4-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1S,5R)-6-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
6-(4-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}piperazin-1-yl)-9H-purine
2-[(1S,5R)-3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(1H-1,2,3-triazol-1-yl)acetamide
(4aR,7aS)-1-ethyl-4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-ylmethyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
thiophen-2-yl(1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-N-(propan-2-yl)pyrimidin-2-amine
1-(4-methylbenzoyl)-4-(2-phenoxyethyl)-1,4-diazepan-5-one
3-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-1-(2-chloro-3,5-difluorophenyl)-3-methylurea
7-(2-methylphenyl)-4-(1,3-thiazol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-(1-methoxypropan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-methoxypropyl)-2-(naphthalen-1-yl)-1H-imidazole
3-{[1-(5-phenyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-yl]methyl}benzamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-yl}ethan-1-ol
N,N,4-trimethyl-5-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]pyrimidin-2-amine
{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[3-(1H-pyrazol-1-yl)propyl]amine
4-{[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzoic acid
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-chlorophenyl)methyl]-N-cyclopropylpyrrolidine-2-carboxamide
N-(dimethyl-1,2-oxazol-4-yl)-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
4-({4-[2-hydroxy-3-(4-hydroxypiperidin-1-yl)propoxy]-3-methoxyphenyl}methyl)piperazin-2-one
N-(dimethyl-1,2-oxazol-4-yl)-4-oxo-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
6-(4-ethylpiperazine-1-carbonyl)-5-methyl-N-[1-(thiophen-2-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
methyl[(2-methyl-1,3-thiazol-4-yl)methyl]{[5-(oxan-2-yl)thiophen-2-yl]methyl}amine
4-methyl-5-(1-methyl-1H-pyrazol-3-yl)-N-[(3,4,5-trifluorophenyl)methyl]-1,3-thiazol-2-amine
[(2S,4R)-4-(dimethylamino)-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-2-yl]methanol
7-(2-methoxyacetamido)-1-methyl-2-(pyridin-3-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(1R,2R,6S,7S)-N-[3-fluoro-5-(trifluoromethyl)phenyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
N,1-dimethyl-6-propyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
4-[5-(3,3-dimethylbutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,6-dimethylquinoline-3-carboxamide
13-(4-chloro-1-methyl-1H-indazol-3-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
N-benzyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-benzofuran-3-carboxamide
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
9-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
1'-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]
N-[2-(3-fluorophenyl)ethyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
2-methyl-9-(piperidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[(dimethylcarbamoyl)amino]phenyl}-2-(thiomorpholin-4-yl)acetic acid
N-[3-fluoro-5-(trifluoromethyl)phenyl]-3-(hydroxymethyl)piperidine-1-carboxamide
N-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-(1,3-thiazol-2-yl)piperidine
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
1-(2-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}-2-oxoethyl)pyrrolidin-2-one
1-cyclohexyl-3-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide