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3-{1-[1-(4-fluorobenzenesulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
2-{1-[4-(3-hydroxy-3-methylbutyl)phenyl]-N-methylformamido}-N,2-dimethylpropanamide
7-(cyclopropylmethyl)-2-(2-propoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
methyl 8-[(3-hydroxy-4-methoxyphenyl)methyl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
1-{3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]morpholin-4-yl}-3-(4H-1,2,4-triazol-4-yl)propan-1-one
ethyl 4-{5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-amido}piperidine-1-carboxylate
1-cyclopropanecarbonyl-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-6-ol
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}acetamide
N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-(2-{[(9H-purin-6-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
2-methoxy-N-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
4-(4-ethylpiperazine-1-carbonyl)-N-[(4-methylphenyl)methyl]aniline
1-{3-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}azepan-2-one
methyl 6-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}pyridine-2-carboxylate
N-({7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,5-dimethylfuran-3-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-amine
3-methoxy-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-methylphenyl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidin-3-ol
ethyl 2-{[3-(2-{[(2-fluorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]amino}acetate
1-(2-chloro-4-fluoro-5-methylphenyl)-3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine
2-{4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]piperidin-1-yl}acetamide
(4aR,6R,8aS)-2-(furan-2-carbonyl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
2-acetyl-8-(2-methylquinolin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-fluoro-3-hydroxy-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylbenzamide
3-[({2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}amino)methyl]piperidin-3-ol
(2R,6R)-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
8-{[5-(dimethylcarbamoyl)furan-2-yl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N,1-dimethyl-N-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
3-[5-(5-chloro-2-methoxybenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-2-(pyridin-3-yl)acetamide
1-(cyclopropylmethyl)-N-ethyl-5-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
ethyl 2-[1-(thiophene-3-carbonyl)piperidin-2-yl]acetate
6-{1-[(2,4-dimethoxy-3-methylphenyl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
2-chloro-4-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)phenol
4-[(2-methylpyridin-3-yl)oxy]-1-(morpholine-4-carbonyl)piperidine-4-carboxylic acid
6-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
N-[2-(2-fluorophenyl)ethyl]-1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
(1,4-dioxan-2-ylmethyl)(1H-indol-7-ylmethyl)methylamine
(3S,4S)-4-({[(6-methylpyridin-2-yl)methyl]amino}methyl)piperidin-3-ol
N-(1-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1H-indol-3-yl}propan-2-yl)acetamide
2-ethyl-5-{2-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-2-oxoethyl}-6-methyl-3,4-dihydropyrimidin-4-one
N-[(3R,4R)-3-hydroxy-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl]pyridine-2-carboxamide
3-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1-(propan-2-yl)pyrrolidine
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-5-methanesulfonyl-N,2-dimethylpyrimidin-4-amine
N-(1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-1-oxopropan-2-yl)propanamide