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N-[2-(4-ethylphenoxy)ethyl]-N-methyl-3-(N-methylmethanesulfonamido)propanamide
N-{[1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-cyclopropyl-4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(1,3-thiazol-2-ylmethyl)benzamide
3-(4-methoxyphenyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-phenylpropanamide
3-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propanamide
3-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]pyridine
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-2-methylpropanamide
1-(3-chloro-4-methoxyphenyl)-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
4-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-2-methoxypyridine
5-(2-chloro-4-fluorophenoxymethyl)-3-[(2R,5R)-2,5-dimethylpyrrolidine-1-carbonyl]-1,2-oxazole
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
6-[(3,5-dimethoxyphenyl)methoxy]-1-(propan-2-yl)-4-(pyridine-4-carbonyl)-1,4-diazepan-2-one
2-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-phenylacetic acid
5-methyl-3-(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-2-yl)-1,2-oxazole
2-{methyl[(4-methyl-5-{1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amino}ethan-1-ol
N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
1-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-[methyl(phenyl)amino]ethan-1-one
2-[5-(2-ethylpyrimidine-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1H-1,3-benzodiazole
(2R,3R,6R)-5-(ethanesulfonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
2-amino-6-(2-methylpropyl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}pyrimidine-4-carboxamide
1-{2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-3,3-dimethylurea
(1S,5R)-6-[(5-ethylpyridin-2-yl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N4,N4,5-trimethyl-N2-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]pyrimidine-2,4-diamine
3-(pyridin-4-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-({1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-3,5-dimethoxybenzamide
N-[(3R,4S)-1-(3-cyanopyridin-2-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
(1S,5R)-6-(cyclopropylmethyl)-3-(4-methylquinolin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(3-chlorophenyl)ethyl]-4-{[(2-methyl-1H-imidazol-4-yl)methyl]amino}pyrrolidin-2-one
N-{2-[7-(2-cyclohexylethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}acetamide
2-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-3-(1H-pyrazol-1-yl)propanamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-ethyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-methyl-1,3-oxazole-5-carboxamide
2,6-dimethoxy-3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)pyridine
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-(2,3-dimethylphenyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxamide
1-{2-oxo-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-methoxy-2-({4-[5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenol
3-[(2-carbamoylmorpholin-4-yl)methyl]benzoic acid
1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-4-(2-methylphenoxy)piperidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-{8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}ethan-1-one
4-(1-butyl-1H-imidazol-2-yl)-1-(2-methylbenzoyl)piperidine
ethyl 1-(prop-2-ene-1-sulfonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
4-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]pyridine
ethyl 4-[(4-chlorophenyl)methyl]-1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
1-(3-methylpyridin-4-yl)-1H-1,3-benzodiazole