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1-(4-acetyl-4-phenylpiperidin-1-yl)-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
N-[(3R,4S)-4-cyclopropyl-1-(diethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-[3-(2-methoxyphenoxy)propyl]-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[4-(ethylsulfanyl)phenyl]urea
2-ethoxy-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
6-({1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)-3-ethyl-3H-imidazo[4,5-b]pyridin-2-amine
N-methyl-4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-N-[2-(pyridin-2-yl)ethyl]pyrimidin-2-amine
N-[(3S,4R)-1-[3-(2-methoxyphenyl)propanoyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
2-(2-{[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenoxy)ethan-1-ol
1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
(3R,4S)-4-{4-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
N-{[7-(1-benzofuran-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2,5-dimethylfuran-3-carboxamide
[(3-chlorophenyl)methyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
(3R,5R)-1-[(3,4-dimethoxyphenyl)methyl]-N-(oxolan-2-ylmethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
5-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)pyridine-2-carbonitrile
1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}-4-(pyridin-3-yl)piperazine
2-{5-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methylacetamide
3,6-dimethyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
6-{[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methyl-1,2,3,4-tetrahydroquinoline
3-{[(4aS,7aR)-4-(cyclopropylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
4-sulfamoyl-N-(thiophen-3-ylmethyl)benzamide
(2S,4S)-4-amino-N,N-diethyl-1-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)pyrrolidine-2-carboxamide
2-(5-ethyl-1-benzofuran-3-yl)-1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]ethan-1-one
methyl 4-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)piperazine-1-carboxylate
7-{2-[(3-methylpyridin-4-yl)amino]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N-[(6-methylpyridin-2-yl)methyl]-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
N-(2-methoxyethyl)-3-{[1-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidin-4-yl]oxy}benzamide
N-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
3-(2,4-dimethylbenzoyl)-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
3-({2-[4-(hydroxymethyl)piperidin-1-yl]ethyl}carbamoyl)-5-methoxybenzoic acid
(3S)-N,N-dimethyl-1-[4-(methylsulfanyl)benzoyl]azepan-3-amine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-benzoyl-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-2-[(2-methoxyethyl)(methyl)amino]acetamide
1-(azepan-1-yl)-3-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}propan-2-ol
2-[2-(4-fluorophenyl)ethyl]-4-[4-(2-methyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[(4-methyl-1H-imidazol-5-yl)methyl]-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)cyclopentanamine
(1R,5R)-3-(3,4-difluorobenzoyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[7-chloro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)thiophene-2-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-{1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-imidazol-2-yl}-N,N-dimethylpyrimidin-2-amine
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
(3aS,6aS)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-octahydropyrrolo[2,3-c]pyrrole
3-hydroxy-1-(2-methoxyethyl)-3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}piperidin-2-one
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
8-(3-propyl-1H-pyrazole-5-carbonyl)-1-oxa-8-azaspiro[4.5]decane
N-[(4-methoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)oxane-2-carboxamide
3,5-difluoro-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)pyridine-2-carboxamide