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N,1-dimethyl-6-propyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[4-(1-hydroxy-3-phenylpropyl)piperidine-1-carbonyl]phenol
1-{2-[1-(2-fluoro-6-methoxybenzoyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
benzyl N-[1-(2,4-dimethylpyrimidine-5-carbonyl)pyrrolidin-3-yl]carbamate
5-acetyl-N-[1-(thiophen-2-yl)propan-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-{2-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-methylpyrrolidin-2-one
2-(2-chloro-6-fluorophenyl)-2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}acetic acid
ethyl 1-[(2-methyl-1,3-thiazol-5-yl)methyl]-4-(2-phenylethyl)piperidine-4-carboxylate
5-methyl-N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)-3-phenyl-1,2-oxazole-4-carboxamide
1-cyclopropyl-N-(furan-2-ylmethyl)-6-oxo-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
[(3R,4R)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-({1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidin-4-yl}methyl)morpholine
1-cyclopropyl-5-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]piperidin-2-one
3-ethyl-1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)piperazine
methyl 1-[9-methoxy-7-oxo-3-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]piperidine-2-carboxylate
2-(3-methyl-1H-pyrazol-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
4-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}morpholine
4-cyclopentyl-2-(4-methanesulfonylphenyl)pyrimidine
methyl 2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)acetate
2-[({1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
4-benzyl-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidine-4-carboxylic acid
2-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(cyclohex-1-ene-1-carbonyl)piperidine-4-carboxamide
(2E)-1-[3-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(pyridin-3-yl)prop-2-en-1-one
9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[1-(2-methoxyethyl)piperidin-4-yl]-1H-imidazol-1-yl}quinoline
3-(3-fluorophenyl)-5-(thiophene-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2-(4-methylpentyl)morpholine
N-cyclobutyl-3-[(3-hydroxyazetidin-1-yl)sulfonyl]benzamide
2-benzyl-9-(4-methylpiperazine-1-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
7-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-2H-chromen-2-one
2-methyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
(2S,4R)-4-amino-N,N-diethyl-1-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}pyrrolidine-2-carboxamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{3-[2-(4-methylpentyl)morpholin-4-yl]-3-oxopropyl}pyrrolidin-2-one
2-(1,3-thiazol-5-ylmethyl)-2,3-dihydro-1,2-benzothiazol-3-one
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-6-(3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-{3-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyrazine
2-cyclopropanecarbonyl-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-propyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,3-thiazole-4-carboxamide
1-phenyl-N-({1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-3-yl}methyl)methanesulfonamide
N-(2,3-dihydro-1H-inden-2-yl)-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
6-methyl-5-{5-[2-(thiophen-2-yl)-1,3-thiazol-4-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
5-fluoro-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}quinazolin-4-amine
2-[(4-methoxypiperidin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
1-methyl-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperazine-2-carboxylic acid