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6-methyl-5-{2-oxo-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(2,4-dioxoimidazolidin-1-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}benzamide
1-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
3-(2-{[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}ethyl)-1,3-oxazolidin-2-one
2-(2,4-dimethoxyphenyl)-3-(pyrrolidin-1-yl)pyrazine
N-[1-(2-chlorophenyl)cyclopropyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-[(1S,5R)-3-{[6-(dimethylamino)pyridin-3-yl]methyl}-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-[2-(azepan-1-yl)ethyl]-5-[(3-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
7-(5-chloropyridin-2-yl)-4-(pyridazine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(1-{6-[(2-hydroxypropyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
N-{2-[cyclopentyl(methyl)amino]ethyl}-N-methyl-1H-1,2,4-triazole-5-carboxamide
N-{3-[5-(2-aminoethyl)-2-methoxyphenyl]phenyl}acetamide
5-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one
N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
7-(2-methoxyphenyl)-2-(pyrimidin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-1H-indole
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)[2-(pyridin-2-yl)ethyl]amine
2-{1-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}benzoic acid
3-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[1-(2,2-dimethylpropyl)-4-hydroxypiperidin-4-yl]-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[1-(piperidin-1-yl)cyclohexyl]methyl}amine
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(pyrrolidine-1-carbonyl)piperidine
2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-N-(propan-2-yl)acetamide
N-cyclooctyl-2-[4-(cyclopropylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]acetamide
6-ethyl-N,2-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}quinoline-4-carboxamide
5-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1H-1,2,3-benzotriazole
2-(ethylamino)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrimidine-5-carboxamide
5-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,2-oxazole-4-carboxamide
(2S)-N-[4-(3-fluorophenyl)phenyl]-1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidine-2-carboxamide
2-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,2-oxazinane
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2-amino-4-phenylpyrimidine-5-carboxamide
5-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
4-(5-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)-1,5-dimethyl-1H-pyrazole
N-{1-[1-(3-aminopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-tert-butyl-3-(2-methanesulfonylacetamido)-2-methylbenzamide
4-[(4-chlorophenyl)methyl]-1-(6-methoxypyrimidin-4-yl)piperidine-4-carboxylic acid
N-[(3-chloro-2-fluorophenyl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
2-(2,4-difluorophenoxy)-N-[2-(5-methylfuran-2-yl)ethyl]acetamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]ethan-1-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(trifluoromethyl)benzamide
8-(5-propylpyrimidin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
(1H-imidazol-2-ylmethyl)(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amine
2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
1-(3-chlorophenyl)-4-[2-(3-chlorophenyl)acetyl]piperazin-2-one
N-(pyridin-2-ylmethyl)-N-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}cyclopropanamine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-4-(1H-pyrazol-5-yl)benzamide
N-methyl-2-(morpholin-4-yl)-N-(3-phenoxypropyl)-2-(pyridin-3-yl)acetamide
N-[(4-phenyloxan-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-{2-[4-(2,5-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-4-ethylpiperazin-2-one
5-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-3-cyclopropyl-1H-1,2,4-triazole