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2-{ethyl[2-(pyrrolidin-1-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-(2-methoxyphenyl)-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-1H-pyrazole-4-carboxamide
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-2,3-dimethoxybenzamide
2-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
N4-ethyl-N2-[(1-ethyl-1H-imidazol-2-yl)methyl]-N2-methylpyrimidine-2,4-diamine
N-(2-chloro-5-fluorophenyl)-4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carboxamide
4-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]azetidin-3-yl}pyridine
4-[4-(2-methylpropanoyl)piperazin-1-yl]-2-(naphthalen-1-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
9-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(3-methyl-1H-1,2,4-triazol-5-yl)-1-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)piperidine
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}cyclobutan-1-amine
3-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-N,N-dimethylazepan-4-amine
{5-[1-(1,3-benzothiazol-6-yl)-1H-imidazol-2-yl]furan-2-yl}methanol
N-methyl-1-[6-(morpholin-4-yl)pyrimidin-4-yl]pyrrolidine-3-carboxamide
[(3R,4R)-1-[2-methyl-5-(trifluoromethyl)benzoyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
[1-(cyclohex-1-ene-1-carbonyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
1-(4-chloro-1H-pyrazole-3-carbonyl)-3-[2-(2,6-difluorophenyl)ethyl]piperidine
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-benzothiophene-5-carboxamide
2-methyl-8-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[6-methyl-2-(2-methylphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(thiophen-3-yl)acetamide
9-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1H-1,3-benzodiazol-2-yl)-2-{[1-(thiophen-2-yl)propyl]amino}acetamide
(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-3-ol
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
methyl 2-{[1-(1-benzylpiperidin-4-yl)piperidin-3-yl]formamido}acetate
1-(pyrimidin-2-yl)-4-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(pyrimidin-4-ylmethyl)benzamide
N-[(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)methyl]acetamide
6-methoxy-3-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-1-benzofuran-2-carboxamide
ethyl 2-[1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]acetate
1-(2,2-dimethylpropyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-[2-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]benzonitrile
3,4,7-trimethyl-N-[2-(methylsulfamoyl)ethyl]-1H-indole-2-carboxamide
2-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)quinoline
7-(3-chlorophenyl)-N,N-diethyl-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
3-{[(4-cyano-2-fluorophenyl)carbamoyl](methyl)amino}-N-methylbutanamide
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-2-methylimidazo[1,2-a]pyridine-3-carboxamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]pyridine-4-carboxamide
3-(morpholin-4-yl)-1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]propan-1-one
1-[1-(2,5-dimethoxybenzoyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
(1R,5R)-6-(2-chlorobenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]pyrrolidin-2-one
2-{4-[5-(6-methylpyridin-2-yl)-1,2,4-oxadiazol-3-yl]phenyl}ethan-1-ol
(2S)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[(4-methanesulfonylphenyl)methyl]methylamine
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide