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4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
[2-(dimethylamino)ethyl](methyl)[2-(1,3-thiazol-2-yloxy)hex-5-en-1-yl]amine
1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]cyclopropan-1-amine
N-[(2S)-1-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-3-(1H-imidazol-4-yl)-1-oxopropan-2-yl]acetamide
2,8-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]quinoline-3-carboxamide
1-(3,5-dimethoxybenzoyl)-N-(3,4-dimethylphenyl)piperidin-3-amine
1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-{[4-(4-methoxyphenoxy)piperidin-1-yl]methyl}pyridine
N-cyclopropyl-5-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-[(2-hydroxyethyl)({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl})amino]-1λ6-thiolane-1,1-dione
2-[(1-hydroxycyclopentyl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[2-(piperidine-1-carbonyl)phenoxy]-1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidine
8-(2-propoxybenzoyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
2-(2-hydroxyphenoxy)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}acetamide
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
5-fluoro-N4,N4-dimethyl-N2-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}pyrimidine-2,4-diamine
4-phenyl-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
1-propyl-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
N-ethyl-4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
5-[({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)(phenyl)methyl]-1,3,4-thiadiazol-2-amine
2-[5-(4-cyanophenyl)-4-phenyl-1H-imidazol-1-yl]-N-(propan-2-yl)acetamide
1-{[3-(difluoromethoxy)phenyl]methyl}-4-ethyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-1-(propan-2-yl)-1H-pyrazole
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(2-fluoro-5-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]acetamide
1-[(3-methoxyphenyl)methyl]-4-(pyrrolidin-3-ylmethyl)piperazin-2-one
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(pyrrolidin-1-yl)propyl]-1,3-oxazole-4-carboxamide
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aR,7aS)-1-(2-methoxyacetyl)-4-(3-methyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aR,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-(thiophene-2-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N2-[1-(2-fluorophenyl)piperidin-4-yl]-N1-(pyridin-3-yl)ethane-1,2-diamine
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[4-(methoxymethyl)piperidin-1-yl]methyl}piperidin-2-one
1-[4-(furan-2-yl)phenyl]-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}piperidin-4-amine
3-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
8-(5-methyl-1H-indole-2-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-1-methylpiperazin-2-one
5-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-2-ethylpyrimidine
N-[2-(1H-imidazol-4-yl)ethyl]-2,3,5,6-tetramethylbenzamide
3-[(4-methoxyphenyl)methyl]-1-methyl-8-[(3-phenoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
ethyl 1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-5-({[(5-methylfuran-2-yl)methyl]amino}methyl)-1H-pyrazole-4-carboxylate
3-methyl-8-{7-methylthieno[3,2-d]pyrimidin-4-yl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,2,6-trimethylquinoline-4-carboxamide
8-[2-(benzyloxy)ethyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-(5-fluoro-2-methoxybenzoyl)-N-(prop-2-en-1-yl)piperidine-1-carboxamide
1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}-3-(pyridin-3-yl)propan-1-one
1-[(3,4-dimethylphenyl)methyl]-4-(1H-pyrrole-3-carbonyl)piperazin-2-one
1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3-(pyrrolidin-1-yl)piperidine