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2-fluoro-6-(isoquinolin-5-yl)benzamide
N-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-4-yl}methanesulfonamide
6-chloro-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]benzamide
N-(1H-imidazol-2-ylmethyl)-2-(1H-indol-3-yl)-N-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
ethyl 1-[3-(cyclopentylcarbamoyl)propanoyl]piperidine-2-carboxylate
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-benzyl-1-{2-oxo-2-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]ethyl}pyrrolidin-2-one
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
{1-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-methanesulfonyl-2-methylpyrimidin-4-amine
6-(4-fluorophenyl)-N-[1-(furan-2-yl)ethyl]-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-cyclopropyl-3-(5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanamide
N2-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-N4,6-dimethylpyrimidine-2,4-diamine
2-[1-(2,2-dimethylpropyl)-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
N-methyl-4-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
N'-cycloheptyl-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]butanediamide
N-(3-{[(4-chlorophenyl)methyl]sulfanyl}propyl)-1-ethyl-1H-pyrazole-3-carboxamide
3-[(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]propan-1-ol
N-{5-[2-fluoro-6-(propan-2-yloxy)phenyl]pyridin-2-yl}methanesulfonamide
(3S,9aR)-8-(3-fluoro-4-methylbenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]butan-2-ol
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
6-cyclopropyl-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]pyrimidin-4-amine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[(2,3-dimethoxyphenyl)methyl]-4-ethyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]formamido}-N,4-dimethylpentanamide
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-phenyl-1,2-oxazol-3-yl)methyl]amine
[(3R,4R)-1-(2,5-dimethylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N-butyl-N-[(2-methylphenyl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
8-(1H-indol-2-ylmethyl)-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-benzothiophene-2-carboxamide
(1S,4S)-2-[2-(methylsulfanyl)phenyl]-5-(quinoline-2-carbonyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
5-(benzylamino)-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1S,5R)-6-(2-methoxypyridine-3-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(1-methoxypropan-2-yl)amine
2-{[4-(1-benzofuran-2-yl)phenyl]methoxy}ethan-1-amine
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(4-ethoxyphenyl)-1-(oxan-4-ylmethyl)-1H-imidazole
N-methyl-3-{1-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]piperidin-3-yl}-N-(1-methylpiperidin-4-yl)propanamide
3-(1H-1,2,3-benzotriazol-1-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}propanamide
ethyl 4-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-3-yl}piperazine-1-carboxylate
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-(4-propanoylphenoxy)acetamide
2-benzyl-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1,3-thiazole-4-carboxamide
2-(2,3-dihydro-1H-isoindol-2-yl)-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
8-(8-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N-(1-{7-[(9-ethyl-9H-carbazol-3-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(quinazolin-2-yl)piperazin-1-yl]propan-1-one
1-(cyclopropylmethyl)-N-methyl-5-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide