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N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[2-(trifluoromethyl)phenyl]methyl}amine
2-(2H-1,3-benzodioxol-5-yloxy)-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
(2R,4S)-4-hydroxy-1-(2-methoxyquinoline-4-carbonyl)piperidine-2-carboxylic acid
N-(2-methoxyethyl)-1-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
N-[3-(morpholin-4-yl)propyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-({5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}methyl)-2-methylpyridine
6-methoxy-3-methyl-N-propyl-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
2-(2-{[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
6-({5H,6H,7H-cyclopenta[b]pyridin-7-yl}amino)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
6-{2-[(6-methoxypyrimidin-4-yl)amino]ethyl}-2-(pyridin-2-yl)-3,4-dihydropyrimidin-4-one
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-9H-fluorene-9-carboxamide
3-(dimethylamino)-N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}pyrrolidine-1-carboxamide
2-{4-[(2,3-difluorophenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
2-[1-({1-[(5-methylthiophen-2-yl)sulfonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]propan-2-amine
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-(2H-1,3-benzodioxol-5-yl)-2-{methyl[(5-methylfuran-2-yl)methyl]amino}acetic acid
4-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N-methyl-1,3-thiazol-2-amine
2-[(3,5-dimethyl-1-benzofuran-2-yl)formamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
1-(2-methylpropyl)-4-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidin-3-yl)piperidine
N-(2-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)acetamide
2-ethoxy-6-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}phenol
2-amino-2-methyl-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
2-methoxy-5-({methyl[(1-phenylpyrrolidin-3-yl)methyl]carbamoyl}amino)benzamide
2-(2-hydroxyethyl)-8-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(1-ethyl-1H-pyrazol-5-yl)-1-[(4-fluorophenyl)methyl]-1-(3-methoxypropyl)urea
(3R,4S)-1-(3-fluoro-4-methylbenzenesulfonyl)-3,4-dimethylpiperidin-4-ol
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-3-(pyrrolidin-3-yl)benzamide
5-ethyl-2-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrimidin-4-amine
1-[1-(4-cyclopentylpyrimidin-2-yl)piperidin-4-yl]piperidin-4-ol
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
2-(1-ethylpiperidin-4-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]acetamide
(4aS,8aR)-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(pyridin-3-ylmethyl)-4-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyrrolidin-2-one
N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
ethyl 2-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,7-diazaspiro[4.5]decane-7-carboxylate
9-(2,6-difluorobenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]piperazine-2-carboxylic acid
N-(3-chloro-4-methoxyphenyl)-6-(cyclohexylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
2,3,6-trimethyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}quinoline-4-carboxamide
5-methoxy-N-methyl-4-oxo-N-[1-(2-phenylethyl)piperidin-3-yl]-1,4-dihydropyridine-2-carboxamide
2,5-dimethyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}benzamide
3-(4-fluorophenoxymethyl)-1-(1-methyl-1H-pyrazole-3-carbonyl)piperidine
1-(6-methylpyridine-2-carbonyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
4-({4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)pyridine
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
(3R,4R)-4-ethyl-1-{2-[(3-fluoro-4-methylphenyl)methyl]benzoyl}piperidine-3,4-diol
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-(2-phenylpropan-2-yl)acetamide