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(3aR,5R,6S,7aS)-2-(1-propyl-1H-pyrazole-5-carbonyl)-octahydro-1H-isoindole-5,6-diol
3-{[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}-2,2-dimethylpropan-1-ol
2-(dimethyl-1,2-oxazol-4-yl)-N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}acetamide
3-(1H-1,3-benzodiazol-1-yl)-N-[(4-phenyloxan-4-yl)methyl]propanamide
({5-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-[(1-benzylpyrrolidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
N-[(3S,4R)-4-propyl-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]acetamide
4-[(3-chlorophenyl)methyl]-1-[(5-methylthiophen-2-yl)methyl]-1,4-diazepan-5-one
5-(5-cyanothiophen-2-yl)-N-(2-methoxyethyl)furan-2-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
N2-[1-(furan-2-carbonyl)piperidin-3-yl]-N4-methylpyrimidine-2,4-diamine
8-(1-benzothiophene-2-carbonyl)-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
(1S,5R)-3-(4-chlorobenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3R,4S)-4-cyclopropyl-1-(1-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]methanesulfonamide
4-[(3-methoxyphenyl)methyl]-1-(9-methyl-9H-carbazole-3-carbonyl)-1,4-diazepan-5-one
3-(4-chloro-1H-pyrazol-1-yl)-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
8-chloro-2-{[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}quinoline
5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[(1S,3S,3aR,6aS)-3-(hydroxymethyl)-5-methyl-3-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]-3-methoxyphenol
3-({4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]acetamide
4-[3-(3,4-difluorophenyl)-5-(1-methylpyrrolidin-3-yl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
(4aS,7aR)-1-(3-hydroxy-4-methoxybenzoyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
4-[(2S)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-2-methylquinoline
[(3R,4R)-1-[(3-fluoro-5-methylphenyl)methyl]-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
4-(2-methoxyphenyl)-2-methyl-1-(2-methyl-1,3-thiazole-4-carbonyl)piperazine
9-[(2-ethylpyrimidin-5-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methoxy-8-[(2E)-3-phenylprop-2-en-1-yl]-1,8-diazaspiro[4.5]decan-2-one
3-chloro-4-({1-[(2,6-difluorophenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
3-(2-methoxyethyl)-5-(2-methyl-1-benzofuran-5-yl)-1,2,4-oxadiazole
7-(2-butoxybenzoyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[4-(1H-indol-4-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]-3-methylbutanamide
2-ethyl-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}pyrimidine-5-carboxamide
1-(4,6-dimethylquinazolin-2-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
4-ethyl-1-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
8-(4-amino-5-methylpyrimidin-2-yl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,4S)-2-(2-chlorophenyl)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-4-sulfamoylbenzamide
(1R,5S,6S)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-3-azabicyclo[3.1.0]hexane
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
3-{1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]azetidin-3-yl}pyridine
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-ethylpyrimidine-5-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]propanamide
2-{5-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-methanesulfonylpropan-1-one
3-amino-N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}benzamide
2-chloro-N-(1-cyclopropanecarbonylpiperidin-3-yl)-5-methylbenzamide
N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-(piperidin-1-ylmethyl)benzamide