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N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
1-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)azepan-4-amine
4-(5,8-dimethoxy-4-methylquinolin-2-yl)-1-methylpiperazine-2-carboxylic acid
(2S,3R)-2-amino-3-hydroxy-1-[5-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butan-1-one
1-[2-(4-chlorophenyl)ethyl]-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
2-cyclopentyl-9-(dimethyl-1,3-oxazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(6-methoxypyridin-2-yl)-2-{[methyl(propan-2-yl)amino]methyl}phenol
1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-4-(1H-1,2,3-triazole-5-carbonyl)-1,4-diazepan-6-ol
1-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
N-methyl-5-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
(4S)-1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3,3,4-trimethylpiperidin-4-ol
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N,1-dimethyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
1-{3-azaspiro[5.5]undecan-9-yl}-4-phenylpiperidine-4-carbonitrile
1-[benzyl(methyl)amino]-3-[4-({[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
methyl 4-({3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)benzoate
(3aR,6aR)-2-[6-amino-2-(morpholin-4-yl)pyrimidin-4-yl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-cyclohexyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-3-ol
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-6-(morpholine-4-carbonyl)pyrazin-2-amine
3-{2-[3-(3-methylphenyl)piperidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
4-(1H-1,3-benzodiazol-1-yl)-1-[(3,4-difluorophenyl)methyl]piperidine-4-carboxylic acid
8-fluoro-2-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}quinoline
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]propan-1-one
2-methoxy-1-{3-[3-(pyridin-4-yl)azetidine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-({1-[(ethylcarbamoyl)methyl]piperidin-3-yl}methyl)-3-(trifluoromethyl)benzamide
N-tert-butyl-4-{3-[(2-methoxyethyl)carbamoyl]phenoxy}piperidine-1-carboxamide
4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}-1λ6-thiomorpholine-1,1-dione
1-{4-[4-(thian-4-yl)piperazine-1-carbonyl]thiophen-2-yl}ethan-1-one
(3R,5S)-N-butyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
2-(4-chloro-2-methylphenoxy)-1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
N-{2-[3-(3-methylbutoxy)phenyl]ethyl}-2,7-dioxo-1,3-diazepane-4-carboxamide
1-[3,5-dimethyl-1-(quinolin-3-yl)-1H-pyrazol-4-yl]ethan-1-one
5-[5-(oxolan-2-yl)thiophene-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
N-[2-(dimethylamino)ethyl]-5-(methoxymethyl)-N-[(2-methylphenyl)methyl]furan-2-carboxamide
N-[3-oxo-3-(pyrrolidin-1-yl)propyl]-3-(piperidin-3-yl)benzamide
3-{2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-4-(2-methylpropyl)piperazin-2-one
1-(2-methoxyethyl)-4-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
6-fluoro-2-({[1-(1H-imidazol-1-yl)butan-2-yl]amino}methyl)quinolin-4-ol
4-[hydroxy(pyridin-2-yl)methyl]-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-2-(trifluoromethyl)morpholine
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N-methylbenzamide
1,3-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(pyridin-3-ylmethyl)-1-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-{[(1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-(3,5-dimethylphenyl)piperazin-2-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)piperidin-3-yl]propan-1-ol
(3S,4S)-N,N-diethyl-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-sulfonamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-(oxan-2-ylmethyl)benzamide