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(1S,5R)-3-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(1S,5R)-6-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-chloro-5-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
3-(5-{[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
2-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
4-({3-[3-(diethylamino)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)-1-methylpiperazin-2-one
N-[(3S,4R)-1-(6-methylpyridazin-3-yl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-cyclopropyl-N-[(4-hydroxyphenyl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-[2-methoxy-5-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
3-(4-fluorophenoxymethyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidine
methyl 2-{1-[(2-phenoxyphenyl)carbamoyl]pyrrolidin-3-yl}acetate
2-(2,5-dioxoimidazolidin-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
2-{imidazo[1,2-a]pyridin-3-yl}-7-phenyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{[(3-methoxypropyl)amino]methyl}-4-(pyrimidin-5-yl)phenol
N-[(3S,4R)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N,1,6-trimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
(3R,4S)-1-[3-(morpholin-4-yl)benzoyl]-4-(propan-2-yl)pyrrolidin-3-amine
6-(1,3-benzothiazol-2-ylmethyl)-N-(pyridin-3-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(1-methoxypropan-2-yl)benzamide
5-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}-3-(propan-2-yl)-1,2-oxazole
N-(oxan-2-ylmethyl)-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(1-methyl-1H-indole-4-carbonyl)piperidin-3-yl]methanol
N3-[2-(cyclohex-1-en-1-yl)ethyl]-N5-(1-hydroxypropan-2-yl)-1-[(2-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(5-chloro-2-methoxyphenyl)-3-[(oxolan-2-ylmethyl)amino]propanamide
6-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]-2-methyl-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)thiomorpholine-4-carboxamide
2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-4-(pyridin-3-yl)pyrimidine
2-(2-methoxyphenyl)-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}pyrimidine
4-[2-(piperidine-1-carbonyl)phenoxy]-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine
(4aR,7aS)-1-methyl-4-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4'-(2,2-dimethylpropyl)-1-(pyridin-3-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-3-yloxy)ethan-1-one
N-cyclohexyl-2-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}acetamide
4-[(4-fluorophenyl)methyl]-1-(pyrrolidin-3-ylmethyl)piperidine
2-{2-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
(3R,5S)-N-[3-(morpholin-4-yl)propyl]-1-(2-phenylethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl})amine
3-{1-[ethyl(methyl)sulfamoyl]piperidin-3-yl}benzoic acid
4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}morpholine
N-[2-(2-cyclohexyl-1H-imidazol-1-yl)ethyl]-3-methylpyridin-4-amine
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-decahydro-2,7-naphthyridin-4a-ol
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
2-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-1,3-benzoxazole
3-(5-{[2-(4,5-dimethylfuran-2-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazol-3-yl)pyridine
1-(pyridin-2-ylmethyl)-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
(2S,4S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-[(2,5-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
5-{2-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
methyl 1-({4-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
(4aS,8aR)-6-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one