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3-[(4-fluorophenyl)methyl]-5-methyl-5-(1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
N-(furan-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-4-methylbenzamide
ethyl 1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-{[7-(pyridin-3-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}propanamide
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
N-(carbamoylmethyl)-N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-[2-(2-phenylethoxy)phenyl]-1H-imidazole
3-(cyclopropylsulfamoyl)-5-(2-fluoro-6-methoxyphenyl)benzoic acid
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
{4-benzyl-1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}methanol
1-[(2,3-difluorophenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
4-({[3-(2-methylpropyl)-1,2-oxazol-5-yl]formamido}methyl)benzoic acid
N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)isoquinoline-1-carboxamide
2-(adamantan-1-yl)-4-hydroxy-N-(2-oxopyrrolidin-3-yl)pyrimidine-5-carboxamide
1-{[3-(difluoromethoxy)phenyl]methyl}-4-(2-phenoxyethyl)piperazine
1-(2-fluorophenyl)-N-[(1R)-2-hydroxy-1-phenylethyl]cyclopropane-1-carboxamide
5-fluoro-2-{4-[(4-methanesulfonylphenyl)methyl]piperazin-1-yl}pyrimidine
N-methyl-N-(1-methylpiperidin-4-yl)-3-[(oxolan-3-yl)sulfamoyl]benzamide
N-benzyl-1-(isoquinolin-5-ylmethyl)-N-methylpiperidin-3-amine
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
2-{[(1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[2-(trifluoromethyl)phenyl]urea
1-{2-[5-(furan-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidine
4-[(4-cyclohexyl-1H-1,2,3-triazol-1-yl)methyl]-1-(1H-imidazole-5-carbonyl)piperidine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(2-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-hydroxy-2-phenylethyl)-N-(pyridin-4-ylmethyl)oxane-4-carboxamide
(2S,4R)-1-[(4-methoxy-3-methylphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N,N-dimethylpyrrolidine-2-carboxamide
4-(4-fluorophenyl)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-ol
[4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-1,4-oxazepan-6-yl]methanol
3-(hydroxymethyl)-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-ol
N-(2-chloro-4-fluorophenyl)-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
(2S)-2-amino-3-hydroxy-1-{4-[4-(propan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}propan-1-one
2-(4-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
(2R)-4-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}-2-methylbutan-1-ol
N-[2-(pyridin-4-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N,N-dimethyl-4-oxo-4-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butanamide
4-(1-methyl-1H-imidazol-2-yl)-1-[2-(pyrrolidin-1-yl)benzoyl]piperidine
2-[(1S,5R)-3-[(5-acetylthiophen-3-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
(1S,5R)-6-{[4-(2-methylpropyl)phenyl]methyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(4-ethynylphenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(3R,4R)-1-({4-amino-6-[(3-methylphenyl)amino]-1,3,5-triazin-2-yl}methyl)-4-cyclobutyl-3-methylpiperidin-4-ol
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(4-fluorophenyl)ethan-1-one
5-[1-(2H-1,3-benzodioxole-5-carbonyl)pyrrolidin-2-yl]-3-methyl-1H-1,2,4-triazole
4-{5-[3-(3-chlorophenyl)pyrrolidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(methylamino)-N-propylpyridine-4-carboxamide
3-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-1-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}urea
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-5-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
14-(2-hydroxy-7-methylquinolin-3-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1-(dimethyl-1,2-oxazole-4-carbonyl)-2-(4-fluorophenyl)piperidine
[3-(hydroxymethyl)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-3-yl]methanol