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2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-5-methylpyrazine
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(4-methyl-1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[5-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-2-(thiophen-3-yl)ethan-1-one
1-(2-methoxyacetyl)-N-(1-phenylpiperidin-4-yl)piperidine-4-carboxamide
3-benzyl-4-(5-phenyl-1,2-oxazole-4-carbonyl)piperazin-2-one
N'-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-N-(propan-2-yl)ethanediamide
N-methyl-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-N-(oxan-2-ylmethyl)piperidine-4-carboxamide
1-[2-(4-methoxy-4-phenylpiperidin-1-yl)-2-oxoethyl]imidazolidin-2-one
N-[2-(1H-indol-3-yl)ethyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-({1-[(4-ethynylphenyl)methyl]piperidin-4-yl}methyl)-2-methylpropanamide
2-[1-(oxan-4-yl)piperidine-3-carbonyl]-2,3-dihydro-1H-isoindole
4-(cyclohexylmethyl)-11-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(3-methoxy-4-methylphenyl)propanamide
2-methyl-6-[(1-propyl-1H-imidazol-2-yl)methyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
4-(2-ethylmorpholin-4-yl)-6-methoxypyrimidin-2-amine
4-({2-[4-(pyrrolidin-1-ylmethyl)phenyl]phenyl}methyl)morpholine
1-(3-chloro-2-methylphenyl)-3-cyclopropyl-5-(2-methoxyethyl)-1H-1,2,4-triazole
N-({1-[(3-cyanophenyl)methyl]piperidin-3-yl}methyl)-1-phenylmethanesulfonamide
1-methyl-3-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}urea
1'-(2-methoxy-4-methylbenzoyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-(2-chlorophenoxy)-1-[(2,3-dimethoxyphenyl)methyl]azetidine
1-methyl-4-(1-{5-[(2E)-pent-2-en-3-yl]-4-phenyl-1H-imidazol-1-yl}butan-2-yl)piperazine
(2S)-N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-oxopyrrolidine-2-carboxamide
1-[(1R,5R)-6-[(3,4,5-trimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-({2-[(2-methoxyethyl)(methyl)amino]acetamido}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2,2,3,3-tetramethylcyclopropane-1-carboxamide
5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
1-[4-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)-1,4-diazepan-1-yl]ethan-1-one
3-[(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}furan-2-yl)sulfanyl]-4-methyl-4H-1,2,4-triazole
3-methyl-2-oxo-N-(4-phenyl-1,2,3-thiadiazol-5-yl)-1-oxa-3,7-diazaspiro[4.5]decane-7-carboxamide
3-[4-(morpholin-4-yl)piperidin-1-yl]-5-(naphthalen-1-yl)-1,2,4-triazine
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
2-fluoro-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
7-methoxy-4-methyl-2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}quinazoline
1-(azepan-1-yl)-2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N,N-dimethyl-2-{[2-(pyrimidin-2-ylsulfanyl)acetamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-{4-chloro-2-[1-(3,4-difluorophenyl)-1H-imidazol-2-yl]phenoxy}acetamide
1-(furan-2-yl)-2-[(3R,4R)-3-hydroxy-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-1-yl]ethane-1,2-dione
3-(3-methoxyphenyl)-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-5-carboxamide
8-(5-propylpyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(3-{1-[(3-methylpyridin-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
1-(pentan-3-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethan-1-ol
8-[(3-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-[1-(1-methylpiperidin-4-yl)-4-{[1-(propan-2-yl)-1H-indol-3-yl]methyl}piperazin-2-yl]ethan-1-ol
N,N-dimethyl-3-[2-({[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)phenyl]propanamide
N-methyl-4-{1-oxa-8-azaspiro[4.5]decane-8-sulfonyl}thiophene-2-carboxamide
N-{2-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-N-methylmethanesulfonamide
2-(3,5-dimethyl-4-{3-[(4-methylphenyl)formamido]propanamido}-1H-pyrazol-1-yl)acetic acid