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N-[3-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)carbamoyl}amino)-4-methoxyphenyl]acetamide
1-cyclopropyl-N-[(3R,5S)-5-(ethylcarbamoyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
7-[2-(2-methylphenyl)acetyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
ethyl 3-[6-amino-5-cyano-4-(1-methyl-1H-pyrazol-4-yl)pyridin-2-yl]benzoate
N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)-4-(4H-1,2,4-triazol-4-yl)benzamide
methyl (2S)-2-[(4,6-dimethylpyrimidin-2-yl)amino]-3-(4-hydroxyphenyl)propanoate
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-methyl-3-oxo-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
ethyl 5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(pyridin-3-yl)-1-[2-(thiomorpholin-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2,4-dimethoxy-N-(oxolan-2-ylmethyl)benzamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(5-fluoro-2-methylphenyl)acetamide
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]acetamide
(2S,4R)-4-amino-1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methylpyrrolidine-2-carboxamide
(2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-4-[(2-hydroxyethyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
2-methyl-4-(4-methylphenyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazine
4-(2-hydroxy-4-methylpentanoyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
1-[2-(3-fluorophenyl)ethyl]-5-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]piperidin-2-one
3-(3-phenyl-1H-pyrazol-1-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
methyl 3-(1,3-dimethyl-1H-pyrazole-5-amido)-5-[(2-methylpropanamido)methyl]benzoate
N-[1-(2-phenylethyl)piperidin-3-yl]quinoxaline-5-carboxamide
4-{4-[(2-fluoro-3-methoxyphenyl)methyl]piperazin-1-yl}-2,6-dimethoxypyrimidine
{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[1-(pyridin-4-yl)propyl]amine
methyl N-{[(2S,4S)-1-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-4-fluoropyrrolidin-2-yl]methyl}carbamate
6-(2,5-dimethylphenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{[3-(pyridin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylcyclopent-1-ene-1-carboxamide
1-[2-(3-hydroxy-4-methoxyphenyl)ethyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]furan-3-carboxamide
methyl 3-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]benzoate
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-4-methyl-1H-imidazole-5-carboxamide
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(3-fluorophenoxy)ethan-1-one
3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-3-yl}benzoic acid
2-[4-(2-chlorophenyl)-3-oxopiperazin-1-yl]propanamide
N,N-dimethyl-6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridazin-3-amine
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]oxane-4-carboxamide
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-6,7-dimethoxy-4-methylquinoline
N-(2-cyclopentylethyl)-2-(methylsulfanyl)pyridine-3-carboxamide
9-ethyl-3-({4-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)-9H-carbazole
3-({[(2,3-difluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
methyl 3-(2-chlorobenzamido)-5-[(pyridin-3-ylformamido)methyl]benzoate
1-cyclopentyl-6-oxo-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidine-3-carboxamide
(2R,3R)-1'-(2-amino-6-hydroxypyrimidin-4-yl)-3-(1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(5-methylpyrazin-2-yl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
3-fluoro-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
4-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]-N-(2-phenylethyl)benzamide
7-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
1-[(1-{6-[(2-hydroxyethyl)(methyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
5-[1-(3-chlorophenoxy)ethyl]-3-methyl-1H-1,2,4-triazole
6-[({[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}amino)methyl]-1,4-oxazepan-6-ol
3-acetyl-N-[(4-methoxyphenyl)methyl]-N-propylbenzamide