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2-{ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}-2-(4-methoxy-3,5-dimethylphenyl)acetic acid
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[2-(methylsulfanyl)acetyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-methyl-4-{octahydro-1H-pyrido[1,2-a]piperazin-2-yl}-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidine
4-fluoro-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-3-methylbenzamide
4-[5-cyclopropyl-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]benzonitrile
[(3R,4R)-1-(3,4-difluorobenzoyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
3-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-N,N-dimethylpyrazin-2-amine
5-ethyl-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidin-2-amine
N-cyclopropyl-4-methoxy-2-({1-[3-(methylsulfanyl)propyl]piperidin-4-yl}oxy)benzamide
4-{1-[3-(pyridin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]propan-2-yl}morpholine
9-[(4-ethoxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(2-methyl-1H-imidazol-4-yl)methyl]amine
1-(4-cyano-2-fluorophenyl)-3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]urea
(4aS,7aR)-1-(cyclohexylmethyl)-4-[2-(dimethylamino)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-chloro-5-acetamido-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}benzamide
5-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine-2-carbonitrile
1-(3-chlorophenyl)-4-[2-(3-hydroxypiperidin-1-yl)acetyl]piperazin-2-one
11-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
N-butyl-5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-cyclopropyl-3-{[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]sulfamoyl}benzamide
1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-(3-{4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}propyl)pyrrolidin-2-one
1-[4-(hydroxymethyl)benzoyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
3-[(2-methyl-1H-imidazol-1-yl)methyl]-1-[4-(pyrrolidin-1-yl)benzoyl]piperidine
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methylbenzamide
(butan-2-yl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)(pyridin-4-ylmethyl)amine
N-[(4-fluorophenyl)methyl]-3-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-4-yl}propanamide
8-{6,8-dioxo-2,7-diazaspiro[4.4]nonan-2-yl}-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
2-{5-[3-(1H-imidazol-1-yl)propyl]-3-methyl-1H-1,2,4-triazol-1-yl}benzoic acid
methyl 5-(1,2,3-thiadiazol-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
dimethyl[(6-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrazin-2-yl)methyl]amine
4-hydroxy-N-(isoquinolin-5-ylmethyl)-N-methyl-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
2-(2-{[3-(4-methylphenoxymethyl)piperidin-1-yl]methyl}phenoxy)acetic acid
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N,2-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}propanamide
1-[3-oxo-3-(pyrrolidin-1-yl)propyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
3-[(4aR,7aS)-4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-[(3S,4R)-1-[2-(1,2-benzoxazol-3-yl)acetyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
(2-{[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]oxy}ethyl)dimethylamine
3-[(2R,3R,6R)-5-(4-hydroxybenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-(2-hydroxyethyl)-8-{7-methylthieno[3,2-d]pyrimidin-4-yl}-2,8-diazaspiro[5.5]undecan-3-one
2-(2-aminoethyl)-5,6-dimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}thieno[2,3-d]pyrimidin-4-amine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}pyrazine-2-carboxamide
2-{[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]methyl}-4-methyl-5,6,7,8-tetrahydroquinazoline
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-1,4-diazepan-2-one
(2R,3R)-3-{[(3-chlorophenyl)methyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
[2-({4-[(4-methyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
2-(2-{[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
5-methanesulfonyl-1'-(5-methyl-1,3-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)-1-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-2-one
5-cyclopropanecarbonyl-1'-(quinolin-4-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]