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4-[(dimethylamino)methyl]-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]benzamide
2-acetyl-8-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-methylpyrimidin-2-yl)piperazin-2-one
cyclohexyl({4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl})methanol
2-[(3,4-difluorophenyl)methyl]-8-(1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-[(3-oxo-1,4-diazepan-1-yl)methyl]-N-[2-(propan-2-yloxy)phenyl]benzamide
1-(2,3-dihydro-1H-isoindol-2-yl)-2-{4-[2-(pyridin-2-yl)acetyl]morpholin-3-yl}ethan-1-one
6-amino-1-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)hexan-1-one
N-(1-{7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
1-[cyclohexyl(methyl)amino]-3-[2-({[2-(1,3-thiazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-methyl-N-[2-(methylsulfanyl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
methyl (2S,4R)-1-({3-[(2,6-dimethylphenyl)carbamoyl]phenyl}methyl)-4-hydroxypyrrolidine-2-carboxylate
3-{2-[methyl(2-phenylethyl)amino]ethyl}-8-(1H-pyrazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-fluoro-N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N,1,3-trimethyl-N-[3-(oxolan-2-yl)propyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-{1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-[2-(3-methoxyphenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
1-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}-4-(pyrrolidin-1-yl)piperidine
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-(3,4-dimethoxyphenyl)-1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-amine
ethyl 1-(2-methylpropyl)-5-{spiro[2.5]octane-1-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-ethoxy-5-(2-{[2-(1H-imidazol-4-yl)ethyl]amino}pyrimidin-4-yl)benzoic acid
N-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
N-butyl-2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methylacetamide
N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-[(2E)-2-methylbut-2-en-1-yl]-3,4-dihydro-2H-1-benzopyran-3-amine
2-cyclobutyl-N-[(3R,4S)-4-cyclopropyl-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]acetamide
4-(2-chloro-5-fluorobenzoyl)-1-(2-methylphenyl)piperazin-2-one
4-hydroxy-N-(oxan-4-yl)-2-phenylpyrimidine-5-carboxamide
N-[3-(dimethylamino)propyl]-1-(2,8-dimethylquinoline-3-carbonyl)-N-methylpiperidin-3-amine
2-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)-4-methylphenol
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-3-(1H-pyrazol-1-yl)propanamide
(4aS,7aR)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
2-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino}pyridine-3-carbonitrile
(3S,4S)-3-({[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-4-hydroxy-1λ6-thiolane-1,1-dione
2-(azocan-1-yl)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}acetamide
3-(diethylamino)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
7-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(azetidine-1-sulfonyl)-N-{3-[ethyl(methyl)amino]butyl}benzamide
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-7-(methylsulfanyl)-3-{[(pyridin-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
methyl (1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxylate
3-(3-chloro-1,2-oxazol-5-yl)-1-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-1-one
(1S,5R)-6-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(2-aminoethyl)-N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
9-{2-[ethyl(methyl)amino]propanoyl}-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-methoxy-1-[3-(2-methylphenoxy)azetidin-1-yl]hexan-1-one
3-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea
methyl 5-[(1-ethylpiperidin-4-yl)amino]-3-(furan-2-amido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2S,4S)-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide