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1-methyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(ethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
5-{[(2,6-difluorophenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2S,4S,5R)-5-(2-chlorophenyl)-1,2-dimethyl-4-[(pyridin-2-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-oxo-3,4-dihydroquinazoline-2-carboxamide
2-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}-1,3-thiazole-4-carboxamide
(1S,5R)-6-(2-methoxypyridine-4-carbonyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-[ethyl(methyl)amino]acetamide
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
(4aR,8aS)-6-[(3-methylphenyl)methyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
7-cyclopentyl-2-(5-propyl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-{1-[4-(dimethylamino)phenyl]propan-2-yl}-2-(1-ethylpiperidin-4-yl)acetamide
methyl 4-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
1-methyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(2-amino-6-methylpyrimidin-4-yl)-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-(ethylsulfanyl)-N-[(1R,3S)-3-(pyrrolidine-1-carbonyl)cyclopentyl]thiophene-2-carboxamide
4-[1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-3-carbonyl]piperazine-1-carbaldehyde
N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
[4-fluoro-3-(5-methyl-1H-indol-3-yl)phenyl]methanamine
N-[(2,5-dimethoxyphenyl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
6-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,3-benzothiazole
(1R,3S,5S)-8-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)-8-azabicyclo[3.2.1]octan-3-ol
(3S,4R)-1-(4-ethoxybenzoyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
4-{[3-(2-aminoethyl)phenyl]methyl}-1-(3-chlorophenyl)piperazin-2-one
3-{[4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine
(3S,4R)-1-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-[2-(2-methoxyphenyl)ethyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-[3-(1,3-thiazole-2-carbonyl)pyridin-2-yl]-1,4-diazepan-6-ol
(benzylsulfamoyl)(methyl)(quinoxalin-2-ylmethyl)amine
N-methyl-N-{1-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}cyclohexanamine
N-({1-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)thiophene-2-carboxamide
(4S,4aS,8aS)-1-{imidazo[1,2-a]pyridine-2-carbonyl}-4-phenyl-decahydroquinolin-4-ol
(2S,4R)-1-[3-(cyclopentylcarbamoyl)propanoyl]-4-(dimethylamino)pyrrolidine-2-carboxylic acid
1-[benzyl(methyl)amino]-3-(5-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
2-[(isoquinolin-5-yloxy)methyl]-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
(4aS,7aR)-1-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-chloro-N,6-dimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[3-(4-methoxyphenyl)propyl]-6-(1,2,3,6-tetrahydropyridin-1-yl)pyridine-3-carboxamide
1-(2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl](methyl)amino}ethyl)piperidin-2-one
N3-butyl-1-cyclohexyl-N5-[3-(dimethylamino)-2,2-dimethylpropyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
2-(4-{[3-(difluoromethoxy)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(1-methyl-1H-pyrazol-4-yl)propanamide
N-[4-(3-fluorophenyl)phenyl]-2-(methoxymethyl)piperidine-1-carboxamide
1-(3-methyl-1H-pyrazole-5-carbonyl)-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N-cyclopropyl-3-{1-[1-(3,5-dimethylphenyl)piperidin-4-yl]piperidin-3-yl}propanamide
2-methoxy-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyrimidine-5-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{2-[2-(5-chlorothiophen-2-yl)-1H-imidazol-1-yl]ethyl}-1,3-oxazolidin-2-one