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6-(oxane-4-carbonyl)-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(2,3-dihydro-1H-inden-4-yl)-3-(2-hydroxyethyl)-3-[(5-methylthiophen-2-yl)methyl]urea
5-methyl-1-(2-phenylphenyl)-4-(1H-pyrazole-3-carbonyl)piperazin-2-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
N,3-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1H-pyrazole-4-carboxamide
(1S,5R)-6-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-({2-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2,2-dimethyl-N-(1-{1-[2-(pyrrolidin-1-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}propan-2-yl)propanamide
4-(1-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}ethyl)morpholine
4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]-1-(1,3-thiazol-2-ylmethyl)piperidine
6-[(9-ethyl-9H-carbazol-3-yl)methyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[(piperidin-4-yl)sulfamoyl]-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
(1S,5R)-6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-[(4-ethoxyphenyl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
8-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[(1-{6-[(4-hydroxybutan-2-yl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
6-cyclopentyl-N,1-dimethyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(4-chlorophenyl)methyl]-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-2,1,3-benzoxadiazole
1-({6-oxo-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)piperidine-4-carboxamide
2-[3-({[(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amino}methyl)phenoxy]acetamide
2-(2-phenylazetidin-1-yl)-N-(5-propyl-1,3,4-thiadiazol-2-yl)acetamide
N-benzyl-N-methyl-1-(pyridin-2-ylmethyl)piperidin-3-amine
3-hydroxy-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
4-{4-[1-(4-chlorophenyl)cyclobutanecarbonyl]piperazin-1-yl}-2-(3,4-dimethoxyphenyl)-2,3-dihydro-1H-isoindole-1,3-dione
8-benzoyl-3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-cyclopentyl-3-[(cyclopentylamino)methyl]-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-[4-fluoro-3-(methylcarbamoyl)phenyl]-4-methanesulfonylpiperazine-1-carboxamide
N-(furan-2-ylmethyl)-N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}-4-methylbenzamide
N,N-diethyl-1-{[1-(pyridin-3-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-[1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
(4aS,7aR)-1-(2-{imidazo[1,2-a]pyridin-3-yl}acetyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4R)-4-amino-1-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
4-{4-[(1S,4S)-5-benzyl-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]phenyl}-2-methylbutan-2-ol
ethyl 3-{[1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
8-benzyl-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}propanamide
3,3-dimethyl-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(morpholin-4-ylmethyl)piperidin-4-ol
(2S,3R)-2-amino-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-3-hydroxybutan-1-one
5-({1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}carbamoyl)-2,1,3-benzoxadiazol-1-ium-1-olate
1-(4-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
5-(2-{[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]amino}pyrimidin-4-yl)-2-ethoxybenzoic acid
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
2-methyl-N-[2-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]propanamide
N-ethyl-5-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]pyrimidin-2-amine
2-({2-[1-(2-chloro-5-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one