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N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2-(3,4,5-trimethoxyphenyl)acetamide
(1R,6S)-9-methyl-3-({5-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,9-diazabicyclo[4.2.1]nonane
1-benzyl-N,N-dimethyl-5-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{3-[(2,4-difluorophenyl)methyl]-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl}methanol
4-{pentacyclo[6.6.6.02,7.09,14.015,20]icosa-2(7),3,5,9(14),10,12,15(20),16,18-nonaen-4-ylmethyl}piperazine-2-carboxylic acid
5-methyl-4-[(4-methyl-1H-imidazol-1-yl)methyl]-2-(2-methylphenyl)-1,3-oxazole
N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
(1S,5R)-6-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(2-methyl-1H-imidazol-4-yl)methyl]-9-oxa-2-azaspiro[5.5]undecane
1-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
N-[1-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-(furan-2-carbonyl)piperidin-4-amine
6-(3-acetylphenyl)-2,4-dimethylpyridine-3-carbonitrile
5-(2,4-difluorophenoxymethyl)-N-(2-methylprop-2-en-1-yl)-1,2-oxazole-3-carboxamide
5-(2-methoxyacetamido)-N,1-dimethyl-2-(pyridin-4-yl)-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
1-(thiomorpholin-4-yl)-3-{2-[({[4-(trifluoromethyl)phenyl]methyl}amino)methyl]phenoxy}propan-2-ol
4-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carbonyl}-4-azatricyclo[4.3.1.13,8]undecane
1-{1-[5-(4-chlorophenyl)-4-methyl-1H-pyrazole-3-carbonyl]azetidin-3-yl}-2-methylpiperidine
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(piperidin-1-yl)ethan-1-one
4-ethoxy-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
5-fluoro-2-(8-methylquinolin-5-yl)phenol
N-benzyl-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(4-methylphthalazin-1-yl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2-[2-(4-fluorophenyl)morpholin-4-yl]-5-methylpyrimidin-4-amine
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(4-fluoro-3-methylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-(2,6-dimethylpyrimidine-4-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-methyl-3-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
3-cyclopropyl-5-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N4-methyl-6-(propan-2-yl)-N4-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidine-2,4-diamine
1-methyl-5-[4-(thian-4-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
4-{7-[(1R,2R)-2-phenylcyclopropanecarbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}morpholine
2-methyl-N-[1-(2-propoxyphenyl)ethyl]-1,3-thiazole-4-carboxamide
N-(2-phenylethyl)-4-{[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]oxy}benzamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(3-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
methyl (1R,3S,3aR,6aS)-1-ethyl-5-methyl-4,6-dioxo-3-[4-(pyridin-2-yl)phenyl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-methyl-4-{1-[(4-phenylphenyl)methyl]pyrrolidin-3-yl}piperazine
N-[4-(methylsulfanyl)phenyl]-4-(pyrrolidin-3-yl)piperazine-1-carboxamide
5,6-dimethoxy-2-{2-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydroisoquinolin-1-one
N-cyclopentyl-N-[(3-ethoxy-4-methoxyphenyl)methyl]-1,3-dimethyl-1H-pyrazole-4-carboxamide
3-hydroxy-N-methyl-N-[(4-phenoxyphenyl)methyl]propanamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-methylpentanamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl){[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
1-{[1-(2-methylpyridin-4-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}azepan-2-one
(1S,3R)-3-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}cyclohexan-1-amine
9-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-(benzyloxy)-4-(1-methylpiperidin-4-yl)-1-(2-methylpropyl)-1,4-diazepan-2-one
2-(1-methyl-1H-pyrazol-3-yl)-1-(1H-1,2,3-triazole-5-carbonyl)piperidine
N-{1-[1-(2-hydroxyethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
ethyl 3-(2-phenoxyethyl)-1-(pyridin-2-ylmethyl)piperidine-3-carboxylate
1-cyclopropyl-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyrrolidin-2-one