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(3S,5R)-5-(cyclopropylcarbamoyl)-1-[(6-methoxynaphthalen-2-yl)methyl]piperidine-3-carboxylic acid
3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-(3-fluorophenyl)piperidine-1-carboxamide
1-(4-cyanopyridin-2-yl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-5-ethyl-N-(pyridin-3-ylmethyl)-1H-pyrrole-2-carboxamide
1-[(3-methoxyphenyl)methyl]-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]piperidin-2-one
(3S,4R)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(hydroxymethyl)piperidin-3-ol
N-[(1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
3-hydroxy-2-{imidazo[2,1-b][1,3]thiazol-6-ylformamido}propanoic acid
1-{1-[2-(4-chloro-2-methylphenoxy)acetyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
methyl[3-(oxolan-2-yl)propyl]{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-cyclopentanecarbonyl-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-[2-(3,4-difluorophenyl)ethyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
1-methyl-4-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
4-ethyl-N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-1,2,3-thiadiazole-5-carboxamide
1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2-(pyrrolidin-1-ylmethyl)piperidine
N-{[5,8-dimethoxy-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2-methyl-1,3-thiazole-4-carboxamide
1,3-dimethyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(3aS,6aR)-5-[(2-chloro-6-fluorophenyl)methyl]-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl 3-[(2-chloro-4-fluorophenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(3-{[(5-methoxy-2-methylphenyl)carbamoyl]amino}propyl)piperidine-4-carboxamide
4-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1-(propan-2-yl)-1H-pyrazole
1-methyl-2-oxo-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1,2-dihydroquinoline-3-carboxamide
1-[2-(1H-pyrrol-1-yl)ethyl]-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
1-[(4-fluoro-3-methylphenyl)methyl]-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
4-{1-[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]propyl}morpholine
2-amino-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-6-(indolizin-2-yl)pyridine-3-carbonitrile
7-propyl-2-[2-(1H-1,2,3,4-tetrazol-1-yl)pyridine-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1-phenylpiperazin-2-one
(2S,4R)-1-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-N-(propan-2-yl)-4-propanamidopyrrolidine-2-carboxamide
(2S,4S)-4-{[(3-chlorophenyl)methyl]amino}-1-{[4-(diethylamino)phenyl]methyl}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
3-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N-cyclohexylpropanamide
2-[4-(6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)acetamide
N-[2-(3-methoxyphenyl)ethyl]-3-(1,2-oxazinan-2-yl)propanamide
4-[(3-ethoxy-2-hydroxypropyl)sulfamoyl]-N-(2-hydroxyethyl)benzamide
2-methoxy-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[1-(piperidin-4-ylmethyl)-1H-1,2,3-triazol-4-yl]methyl}amine
5-chloro-2-(2-phenyl-1H-imidazol-1-yl)pyridine
4-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]phenol
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2,4,6-trimethylbenzamide
N-{[(2S,4S)-1-[benzyl(methyl)sulfamoyl]-4-fluoropyrrolidin-2-yl]methyl}-2-methoxyacetamide
ethyl 1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperidine-3-carboxylate
N-(furan-2-ylmethyl)-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
methyl 4-{5-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-1,2,4-oxadiazol-3-yl}benzoate
7-cyclohexyl-2-(5-fluoro-2-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
5-(2H-1,3-benzodioxol-5-yl)-3-[(4-phenyl-5-propyl-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole