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N-[2-(1H-indol-1-yl)ethyl]-1-methyl-1H-pyrazole-5-carboxamide
4-[(2-fluorophenyl)methyl]-1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-1,4-diazepan-5-one
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-7-oxo-3-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-methyl-N-{2-[3-(propan-2-yloxy)phenyl]ethyl}piperidine-4-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
7-cyclohexyl-2-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-[4-(2H-1,3-benzodioxol-5-yl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(3aR,6aR)-2-methyl-N-[2-(methylsulfamoyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
1-[(3-fluorophenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydropyrimidin-2-one
1-(2-ethoxyethyl)-4-(thiophene-3-carbonyl)-1,4-diazepane-6-carboxylic acid
3,5-dimethyl-N-(thiolan-3-yl)-1,2-oxazole-4-carboxamide
N-(1-{7-[(2,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
1-[(4-methoxy-3-methylphenyl)methyl]-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2,3-dihydro-1-benzofuran-7-carboxamide
2-methyl-N-{[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-(oxane-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperazine
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-6-(2,5-dimethylphenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine
3-[(2,1,3-benzothiadiazol-5-ylmethyl)sulfamoyl]-N,N-dimethylbenzamide
4-amino-1-cycloheptylpyrrolidin-2-one
1-(2-aminopyridine-4-carbonyl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
6-ethyl-4-methyl-2-(pyridin-4-yl)quinoline
2-[(3-chloro-4,5-dimethoxyphenyl)methyl]-9-oxa-2-azaspiro[5.5]undecane
N-{4-chloro-3-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octane-8-carbonyl]phenyl}acetamide
3-tert-butyl-4-(3-cyclohexyl-1H-pyrazol-4-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(2,4-dihydroxyphenyl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
(1S,5R)-6-benzyl-3-(1H-imidazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{[benzyl(methyl)amino]methyl}-N-[(1-methylpiperidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
N-{[7-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(phenylsulfanyl)acetamide
3-[(3R,4S)-1-[(3,4-dimethylphenyl)carbamoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-[9-(2-fluorobenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
2,6-dimethyl-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}quinoline-3-carboxamide
3-(2-{2-azabicyclo[2.2.1]heptan-2-yl}-2-oxoethyl)-3-(2-methoxyphenyl)-1-(3-methoxypropyl)pyrrolidine-2,5-dione
4-[3-(1H-pyrazol-4-yl)benzoyl]-2-(trifluoromethyl)morpholine
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-3,6-dimethyl-1-benzofuran-2-carboxamide
N-[2-(4-fluorophenyl)-1-{1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-4-yl}ethyl]-2-methoxy-N-methylacetamide
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2,6-dimethoxybenzamide
2-(1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol
2-benzyl-N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1,3-thiazole-4-carboxamide
1-{2-hydroxy-5-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenyl}ethan-1-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-N-methylpropanamide
4-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrimidine-5-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)(2,1,3-benzothiadiazol-4-ylmethyl)(pyridin-3-ylmethyl)amine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(morpholine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-{[3-(2-fluorophenoxy)azetidin-1-yl]methyl}quinoline
3-[5-(1-cyclopentanecarbonylpiperidin-4-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amine