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1-[(1-ethylpiperidin-2-yl)methyl]-4-(4-methylphenoxy)piperidine
N,N-diethyl-1-[3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine-3-carboxamide
3-[(dimethylamino)methyl]-1-[4-(1H-pyrazol-3-yl)benzoyl]pyrrolidin-3-ol
N-[(1-{2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-3-yl)methyl]acetamide
2-(methylamino)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
N,N-dimethyl-4-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline
2-{[3-(4-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}-4-methanesulfonylbutanoic acid
1-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
(7R,9aR)-N-cyclohexyl-7-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-{2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
5-(3-benzylpyrrolidine-1-carbonyl)-3-(4-fluorophenyl)-1H-pyrazole
(3aR,6aR)-2-(prop-2-en-1-yl)-5-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(2-phenylethyl)piperidin-3-yl]pyridine-3-carboxamide
N-[2-(1,3-benzothiazol-2-yl)ethyl]-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
8-(furan-2-carbonyl)-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
(3R,5S)-5-(3-fluorophenoxymethyl)-N-[3-(morpholin-4-yl)propyl]-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
N-{3-methyl-1-[7-(quinolin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}furan-2-carboxamide
(7-methyl-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}quinolin-3-yl)methanol
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)acetamide
2-[4-(1-methoxyethyl)phenyl]-5,6-dimethylpyridine-3-carboxamide
methyl 4-{[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}butanoate
2-amino-6-cyclopropyl-4-[2-(ethylsulfanyl)pyrimidin-5-yl]pyridine-3-carbonitrile
2-methyl-8-{1H-pyrazolo[3,4-b]pyridin-4-yl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-methyl-6-(2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}ethyl)pyrimidin-4-ol
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-(6-methoxyhexanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S,4R)-N,N-diethyl-4-(1-methylcyclopropaneamido)-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]propan-1-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}acetamide
(4aS,7aR)-1-(3-cyclopentylpropanoyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(4-methyl-1H-pyrazol-3-yl)piperidine
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-(1-methyl-6-oxopiperidin-3-yl)pyrimidine-5-carboxamide
2-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydrophthalazin-1-one
1-cyano-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}cyclopropane-1-carboxamide
N,N-dimethyl-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]azepan-4-amine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-methoxybutanamide
1-cyclopentyl-4-{4-[2-(propan-2-yloxy)phenyl]-1H-imidazol-2-yl}pyrrolidin-2-one
4-({1-ethyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}methyl)-N,N-dimethylaniline
2-methyl-8-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
5-(cyclohex-3-en-1-yl)-1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
(4-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)methanol
6-(2-hydroxyethyl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[(1S,2R)-2-butylcyclopropanecarbonyl]-4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine
2-amino-4-(3,5-dimethyl-1H-pyrazol-4-yl)-6-(3-hydroxyphenyl)pyridine-3-carbonitrile
3-[1-(4-methoxyphenyl)-1H-1,3-benzodiazol-2-yl]propan-1-ol
2-methoxy-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-phenylethan-1-one
4-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1-methylimidazolidin-2-one