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N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(4-methylphenyl)methyl]piperidin-3-yl}propanamide
N-(3-cyclopentylpropyl)-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
4-(cyclohex-3-en-1-ylmethyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3R,4R)-3,4-dimethyl-1-[6-(4-methylpiperazine-1-carbonyl)pyrazin-2-yl]pyrrolidin-3-ol
N-[(2,4-difluorophenyl)methyl]-5-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-methyl-3-phenoxy-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
1-(1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)-4-(piperidin-1-yl)piperidine
3-{5-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2,2-dimethyloxane-4-carboxamide
N,N-bis(1,3-oxazol-4-ylmethyl)-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-(2-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
methyl 4-{[5-(2,4-difluorophenoxymethyl)-1,2-oxazol-3-yl]formamido}butanoate
N-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
3-[4-(4-ethylpiperazin-1-yl)piperidine-1-carbonyl]-N,N-dimethyl-6-(thiophen-2-yl)pyridin-2-amine
N-ethyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-(3-phenylpropyl)acetamide
N-(oxolan-2-ylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
(4aS,8aR)-6-[(2-aminopyridin-3-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-(2-chloro-5-fluorophenyl)-4-(2,6-dimethylpyridin-4-yl)piperazine-1-carboxamide
4-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}-N-[(3S)-piperidin-3-yl]benzamide
2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[3-(1,3-thiazol-4-yl)phenyl]acetamide
7-(cyclopropylmethyl)-2-[(2-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
methyl 1-ethyl-5-[(4-methoxy-4-methylpentan-2-yl)amino]-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(4-methyl-1,3-oxazole-5-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
5-ethyl-4-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
1-[(diethylcarbamoyl)methyl]-N-[1-(thiophen-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1,4-dihydroquinolin-4-one
N-(1-hydroxypropan-2-yl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
3-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propanamide
2-{1-[(3,4-difluorophenyl)methyl]-4-[(2,5-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide
6-[(3-aminoazepan-1-yl)methyl]-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(1-cyclopropylethyl)-3-methyl-1H-pyrazol-5-yl]-4-(1,3-thiazol-2-yl)piperazine-1-carboxamide
methyl 2-{[(4-methylphenyl)methyl]sulfamoyl}-6-(2-methylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]-1-[(4-methylphenyl)methyl]pyrrolidine-2-carboxamide
1-(2-methoxypyridine-4-carbonyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
1-[5-(3-methylbut-2-en-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]pyrrolidine
(2S,4R)-4-amino-1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2-hydroxyphenyl)methyl]piperidin-3-yl}propanamide
2-(2,4-dichlorophenoxy)-N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}acetamide
4-[(methylsulfanyl)methyl]-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine
5-[methyl(2-phenylethyl)amino]-2-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,3-dihydropyridazin-3-one
2-(3-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenoxy)acetamide
2-methoxy-1-(4-{[2-(trifluoromethoxy)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one
2-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-2-yl)pyridine
[(1-methyl-1H-pyrazol-4-yl)methyl]({[2-(2-methylphenoxy)pyridin-3-yl]methyl})amine
methyl 4-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
6-[2-(3-chlorophenoxy)propanoyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one