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N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
1-{1-[6-(cyclopropylamino)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
N-methyl-1-(2-phenylethyl)-N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
(3R)-1-(2-methanesulfonylethyl)-3,4,4-trimethylpyrrolidin-3-ol
1-[2-(1H-imidazol-4-yl)ethyl]-2-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-imidazole
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-5-[1-(furan-2-ylmethyl)-4-hydroxypiperidin-4-yl]-1-benzofuran-2-carboxamide
5-ethyl-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]thiophene-3-carboxamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-[4-(6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
[1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)piperidin-4-yl]diphenylmethanol
2-ethyl-N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]pyrimidine-5-carboxamide
1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
5-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2,4-dimethyl-1,3-thiazole
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
[(3aS,6aS)-2-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
1-(2-{[ethyl(methyl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)-4-(4-fluorophenyl)butane-1,4-dione
4-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
4-(2-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]formamido}ethyl)benzoic acid
3,5-dimethoxy-N-({1-[2-(2-oxopiperidin-1-yl)acetyl]piperidin-3-yl}methyl)benzamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-6-methoxy-N,1-dimethyl-1H-indole-2-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-[(2S,4R,6S)-2-(4-butoxyphenyl)-6-ethyloxan-4-yl]acetamide
1-cyclohexyl-3-(oxolan-3-yl)-5-[(phenylsulfanyl)methyl]-1H-1,2,4-triazole
6-(2-hydroxyethyl)-N-[1-(methylcarbamoyl)cyclohexyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(2-chloro-4,5-difluorophenyl)-1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]ethan-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}acetamide
methyl (2S,3S)-3-methyl-2-{[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}pentanoate
1-[5-(4-cyclohexylphenyl)-1,2,4-triazin-3-yl]-4-(pyrimidin-2-yl)-1,4-diazepane
1-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(4-methylphenyl)ethan-1-one
N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
[(3R,4R)-1-{[3-methoxy-4-(propan-2-yloxy)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-(2,3-dihydro-1H-inden-2-yl)-4-[(quinoxalin-2-yl)amino]pyrrolidin-2-one
N-[2-hydroxy-2-(pyridin-2-yl)ethyl]-3,5,7-trimethyl-1H-indole-2-carboxamide
4-{4-[(dimethylcarbamoyl)amino]phenyl}-N-methylbenzamide
1-[3-(4-fluorophenoxy)propyl]-4-(5-methyl-1,3,4-oxadiazol-2-yl)piperazine
(1R,5R)-6-(2-amino-6-methylpyrimidine-4-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
N-[(3R,4R)-1-[3-(3-fluorophenyl)propanoyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
3-[(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-3-yl)methyl]benzoic acid
N-[2-(3,4-dimethoxyphenyl)ethyl]-3-[(3S,4R)-4-(dimethylamino)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]propanamide
2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
4-{[2-(2-oxoimidazolidin-1-yl)ethyl]sulfamoyl}-N-propylbenzamide
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
methyl 2-[butyl(methyl)sulfamoyl]-6-[(2,6-difluorophenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-acetyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1H-pyrazole-5-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[3-(2-ethylphenoxy)azetidin-1-yl]ethan-1-one
4-[4-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidin-1-yl]-1λ6-thiane-1,1-dione
4-(3-hydroxy-3-methylbutyl)-N-[2-(1-hydroxycyclopentyl)ethyl]-N-methylbenzamide
3-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]pyridin-2-ol