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5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-3,5-dimethyl-4,5-dihydro-1,2-oxazole
(4aR,8aR)-2-(4-cyclobutyl-6-methylpyrimidin-2-yl)-7-cyclopentanecarbonyl-decahydro-2,7-naphthyridin-4a-ol
6-(2-{[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]amino}ethyl)-2-methylpyrimidin-4-ol
1-methyl-4-{[2-(morpholin-4-yl)quinolin-3-yl]methyl}piperazin-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-propyl-1,3-thiazole-4-carboxamide
diethyl({[1-(1-methylazepane-2-carbonyl)pyrrolidin-2-yl]methyl})amine
({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})amine
8-{6-azaspiro[2.5]octane-1-carbonyl}-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-1-[(5-methyl-1H-pyrazol-3-yl)methyl]piperidine
4-(5,6-dimethylpyrimidin-4-yl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl][(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amine
1-(4-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-1-yl)ethan-1-one
2-({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[(1-ethylcyclobutyl)methyl]-1-(3-methyl-1,2,4-thiadiazol-5-yl)urea
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-(1H-imidazol-2-ylmethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(1H-pyrazol-1-yl)acetamide
3-[2-(azepan-1-yl)-2-oxoethyl]-4-(naphthalen-2-ylmethyl)piperazin-2-one
2-(benzyloxy)-N-[(1-methylpiperidin-4-yl)methyl]acetamide
(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(2E)-3-(3-fluorophenyl)-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)prop-2-enamide
2-amino-N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
4-phenyl-1-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-one
2-(4-methyl-1H-1,3-benzodiazol-2-yl)-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)pyrrolidine-1-carboxamide
1-[2-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
3-(3-fluorophenyl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]propan-1-one
1-{2-[1-cyclohexyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
N-[3,5-difluoro-4-(trifluoromethyl)phenyl]-3-ethylpiperazine-1-carboxamide
5-{[(2,3-dimethoxyphenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-(dimethylamino)-N-[3-(3-methyl-1H-pyrazol-1-yl)propyl]-2-(4-methylphenyl)acetamide
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(2-methoxyethoxy)ethan-1-one
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-2-oxo-4-[4-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepan-6-yl}oxy)acetamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)(thiophen-3-ylmethyl)amine
5-(4-fluorophenyl)-2-methyl-4-{1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl}pyrimidine
5-(2H-1,3-benzodioxol-4-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazole
N-[(2S,4R,6R)-2-(5-chloro-3-methyl-1H-indol-2-yl)-6-(propan-2-yl)oxan-4-yl]acetamide
N-benzyl-N-methyl-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-3-amine
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
1-(2-ethylpyrimidine-5-carbonyl)-N,N-dimethylazepan-4-amine
N-cyclopropyl-1-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
[(3R,4R)-1-(5-methyl-1,3-benzoxazol-2-yl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4-methyl-6-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]pyrimidin-2-amine
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(1,3-thiazol-5-ylmethyl)piperidine-2-carboxamide
1-[(2-ethyl-4-methyl-1,3-oxazol-5-yl)methyl]-4-(pyrrolidin-1-yl)piperidine
8-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]-1-oxa-8-azaspiro[4.6]undecane
N-[3-(3-chlorophenyl)phenyl]-1-(pyridine-2-carbonyl)piperidine-4-carboxamide
(4aS,7aR)-1-(1H-indole-6-carbonyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
14-(5-fluoro-2-methoxyphenyl)-6-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
(5S,9aS,9bS)-2-(3-methoxyphenyl)-5-(4-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one