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1-methyl-4-(3-phenylpropanoyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
9-(3-fluoropyridin-4-yl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-5,6,7,8-tetrahydroquinoline-3-carboxamide
2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-N,N-dimethylacetamide
5-[3-(2-methylphenyl)piperidine-1-carbonyl]pyrazin-2-ol
7-(2,1,3-benzoxadiazol-4-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(4-fluorophenyl)-N-(2-{7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
(1S,5R)-6-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-(2,5-dimethoxyphenyl)-2-{[4-(2-ethoxyphenyl)piperazin-1-yl]methyl}phenol
N3-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-N5-cycloheptyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)benzamide
1-tert-butyl-N-[2-(2,3-dichlorophenyl)ethyl]-5-oxopyrrolidine-3-carboxamide
3-(5-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl)pyridine
4-(hydroxymethyl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]azepan-4-ol
[(4aS,8aR)-6-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
2-{4-cyclopentyl-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(pyrrolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
2-amino-4-(1-methyl-1H-pyrazol-4-yl)-6-(3-propoxyphenyl)pyridine-3-carbonitrile
2-{4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-3-carboxamide
2-(4-{5-cyclopropyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazin-1-yl)phenol
2-cyclopropyl-4-hydroxy-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrimidine-5-carboxamide
2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-3-(4-phenylazepane-1-carbonyl)-1,4-dihydropyridin-4-one
N-[3-(pyridin-3-yloxy)propyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
N,N-dimethyl-6-[3-(1-{[(propan-2-yl)carbamoyl]methyl}-1H-pyrazol-3-yl)phenyl]pyrazine-2-carboxamide
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(pyridin-2-yl)propan-1-one
(2S)-1-acetyl-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]pyrrolidine-2-carboxamide
N4-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine-4,6-diamine
6-methyl-2-{2-[5-methyl-5-(4-methylpent-3-en-1-yl)-2-oxopiperidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
1-(benzenesulfonyl)-4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
2-hydroxy-4-methoxy-N-(3-phenylprop-2-yn-1-yl)-N-propylbenzamide
(3S,9aR)-8-(2,5-difluorobenzoyl)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-({[2-(azocan-1-yl)pyridin-3-yl]methyl}amino)pyrazine-2-carboxamide
3-[(3R,4S)-1-[2-(4-fluoro-3-methylphenyl)acetyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(4-methoxybenzoyl)piperazine
(3S,4S)-4-propyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidine-3-carboxylic acid
8-(3-methyl-5-{[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]methyl}-1H-1,2,4-triazol-1-yl)quinoline
4-{3-[4-(pyridin-4-yl)-1,4-diazepane-1-carbonyl]phenyl}phenol
3-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-{[4-(hydroxymethyl)oxan-4-yl]methyl}urea
2-{2-[1-(quinoline-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
6-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N5-[(2,5-difluorophenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
8-[(4-chlorophenyl)carbamoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-(1H-indazole-3-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N,N,1-trimethyl-3-[4-(1H-pyrazol-5-yl)phenyl]-1H-1,2,4-triazol-5-amine
3-[1-(5-hydroxypyrazine-2-carbonyl)piperidin-3-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-fluoro-5-methoxyphenyl)-2-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}acetic acid
N-[1-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-4-phenylbutanamide
2-[1-(furan-2-ylmethyl)-4-{imidazo[1,2-a]pyridine-2-carbonyl}piperazin-2-yl]ethan-1-ol
3-(1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(3-fluorophenyl)urea