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7-[(2,3-difluorophenyl)methyl]-2-[(5-methylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyridine-3-carboxylic acid
2-(cyclopropylmethyl)-9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
4-chloro-5-({[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amino}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
N-{3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propyl}pyridin-3-amine
N-({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)-N-methylthian-4-amine
3-(3-hydroxy-3-methylbutyl)-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]benzamide
2,2-dimethyl-N-{[1-(quinolin-2-ylmethyl)piperidin-3-yl]methyl}propanamide
N-[(3R,4S)-1-[1-(methoxymethyl)cyclopropanecarbonyl]-4-propylpyrrolidin-3-yl]-5-methyl-1,2,4-oxadiazol-3-amine
2-({[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}methyl)-6-fluorophenol
6-fluoro-2-({[3-(pyrrolidin-1-yl)propyl]amino}methyl)quinolin-4-ol
N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)thiophene-2-sulfonamide
N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
1-[7-(3-chlorophenyl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2,5-dimethoxyphenyl)ethan-1-one
(2R)-2-amino-3-(4-chlorophenyl)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
N-(2-hydroxyethyl)-N-propyl-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]benzoic acid
2-fluoro-N-[3-(morpholin-4-yl)propyl]-5-sulfamoylbenzamide
2-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidine-3-carbonyl}pyridine
5-cyclopropanecarbonyl-1'-(6-methylpyridazin-3-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-amine
1-[3-({3-[(2R,5R)-2,5-dimethylpyrrolidine-1-carbonyl]-1H-pyrazol-5-yl}methoxy)phenyl]ethan-1-one
(3S,9aR)-3-benzyl-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(butan-2-yl)-6-methyl-5-[5-(1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
5-[4-(azepan-1-ylmethyl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(3R,5S)-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-(2-oxo-2-{3-oxo-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-6-yl}ethyl)-1,2-dihydrophthalazin-1-one
4-(1-benzoxepine-4-carbonyl)-3-butyl-1-methylpiperazin-2-one
methyl (2S,4R)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-hydroxypyrrolidine-2-carboxylate
N,2,3,5-tetramethyl-N-(pyrazin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
(4aS,8aR)-6-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
4-(7-chloro-2-methylquinoline-4-carbonyl)-1-phenylpiperazin-2-one
6-(4-methoxyphenyl)-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
4-({2-[3-(morpholin-4-yl)propoxy]phenyl}methyl)morpholine-2-carboxamide
1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-3-(3-methylthiophene-2-carbonyl)piperidine
1-{1-[1-(2,2-diethylcyclopropanecarbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}cyclopentan-1-ol
1-[(5-ethylpyridin-2-yl)methyl]-4-(oxan-4-yl)piperazine
methyl 2-(1-{[3-(furan-2-yl)phenyl]carbamoyl}pyrrolidin-3-yl)acetate
5-[4-(hydroxymethyl)-1,3-thiazol-2-yl]thiophene-2-carboxylic acid
4-(3-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}phenyl)-1H-pyrazole
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-(4-methylphenoxy)ethan-1-one
2-{3-[(2R,5S)-2,5-dimethylpyrrolidine-1-carbonyl]phenyl}-1H-imidazole
2-(3-{[methyl({[2-(pyrrolidin-1-ylmethyl)phenyl]methyl})carbamoyl]amino}phenyl)acetamide
N-(1-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
(3aR,6aS)-5-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
3-(5-methylthiophen-2-yl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-[2-(4-fluorophenoxy)ethyl]-3-methoxy-1,2-dihydropyridin-2-one
1-[1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol