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7-(5-methylthiophen-2-yl)-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(2-fluorophenyl)methyl]-4-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperazin-2-one
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(5-ethylfuran-2-yl)methyl]piperidine
7-(1,3-benzothiazol-2-yl)-4-[2-(pyridin-2-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-(5-hydroxypyrazine-2-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-[(3,5-dimethylphenyl)sulfamoyl]-6-(1-methyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[methyl({[2-(piperidin-1-yl)pyrimidin-5-yl]methyl})amino]-1λ6-thiolane-1,1-dione
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2-(pyridin-4-yl)acetamide
2-amino-3-ethyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-methyl-8-[2-(6-methylpyridin-2-yl)ethyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(2-cyclopropylphenyl)-1-{2-[(3-methylpyridin-2-yl)amino]ethyl}urea
1-(but-3-enoyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
ethyl 5-methyl-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1S,5R)-3-methyl-6-{[3-(5-methylfuran-2-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
4-(3-benzyl-1H-pyrazol-5-yl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-(cyclohexyloxy)-3-[(pyrimidin-4-yl)amino]propan-2-ol
N-cyclobutyl-4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-2-methyl-4-(4-methylphenyl)piperazine
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[4-(hydroxydiphenylmethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-{[4-(aminomethyl)phenyl]methyl}-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
5-chloro-N-methyl-N-(oxolan-2-ylmethyl)-3-phenyl-1H-indole-2-carboxamide
1-acetyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]piperidine-4-carboxamide
(4aS,8aS)-2-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-decahydroisoquinoline
1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}spiro[azepane-4,2'-chromene]
2-ethoxy-6-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenol
3-[1-(2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}acetyl)piperidin-3-yl]benzoic acid
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-(thiophen-2-yl)acetamide
[(1-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl](methyl)amine
ethyl 2-[methyl({8-methyl-2-[methyl(2-phenylethyl)carbamoyl]imidazo[1,2-a]pyridin-3-yl}methyl)amino]acetate
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2-methyl-1H-imidazol-1-yl)ethan-1-one
7-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-4-methoxy-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
3-(3,4-difluorophenyl)-5-(3-fluoro-4-methoxybenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(2S,4S)-N-ethyl-1-(1-propylpiperidin-4-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
4-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-4-oxobutane-1-sulfonamide
(3aR,7aS)-2-[4-methoxy-3-(morpholin-4-yl)benzoyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-(2-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}ethyl)-4-(2-methyl-1,3-thiazole-4-carbonyl)piperazine
5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-1-(4-fluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]butanamide
N-(5-methyl-1,2-oxazol-3-yl)-2-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}acetamide
(1S,6R)-9-(4-propylpyrimidine-5-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-(4-phenylpiperazine-1-carbonyl)piperidin-2-one
5-{[1-(5-chloro-2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2-methyl-3,4-dihydropyrimidin-4-one
1-(3-{4-azaspiro[2.5]octan-4-ylmethyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(propan-2-yl)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
1-(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-phenylpiperidin-4-yl)ethan-1-one
N-({1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}methyl)-2-(1H-pyrazol-1-yl)acetamide