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N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-{2-[cyclopentyl(methyl)amino]ethyl}-N,1-dimethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-benzyl-5-{[2-(4-fluorophenyl)ethyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(7,7-dimethyl-5-{[4-methyl-6-(methylamino)pyrimidin-2-yl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-ol
N-[(2-chlorophenyl)methyl]-N-methyl-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-[4-(1H-pyrazol-5-yl)phenyl]-1-[2-(pyridin-4-yl)acetyl]piperidine-3-carboxamide
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
8-[(2-methoxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(6-chloropyridin-3-yl)-4-hydroxy-4-(pyridin-3-yl)piperidine-1-carboxamide
methyl 4-{[9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoate
methyl 4-[(4-acetyl-4-phenylpiperidin-1-yl)methyl]-1H-pyrazole-3-carboxylate
4-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)morpholine
2-(2-ethoxyphenyl)-1-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1H-imidazole
3,6-dimethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1-benzofuran-2-carboxamide
2-{1-[(5-methylpyrazin-2-yl)methyl]-1H-1,2,3-triazol-4-yl}quinolin-4-ol
6-(isoquinolin-5-yl)-N-methylpyridine-2-carboxamide
1-[(3R,4S)-3-[(6-cyclopropylpyrimidin-4-yl)amino]-4-propylpyrrolidin-1-yl]-2-(methylamino)ethan-1-one
(2S,4R)-4-amino-N-ethyl-1-[(4-ethylpiperazin-1-yl)sulfonyl]pyrrolidine-2-carboxamide
1-(cyclohexylmethyl)-N-[2-(pyridin-3-yloxy)ethyl]-1H-1,2,3-triazole-4-carboxamide
ethyl 2-[9-(2,3-dihydro-1H-inden-2-yl)-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]acetate
({3-methyl-1-[2-(4-methylpiperazin-1-yl)ethyl]-1H-pyrazol-4-yl}methyl)[(2-methylphenyl)methyl]amine
3-{1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
2-[4-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenyl]-6-(methoxymethyl)-3,4-dihydropyrimidin-4-one
5-fluoro-2-(3-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}urea
3-(but-2-yn-1-yl)-5-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
N-({5-[(5-ethylpyridin-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(1H-indol-3-yl)-N-methylpropanamide
[(3R,4R)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-amino-1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
4-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}-5,6,7,8-tetrahydroquinazolin-2-amine
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
(2-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}-2-oxoethyl)urea
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)-1-(thiophen-2-ylmethyl)piperidine
6-chloro-2-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}quinoline
4-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydroquinolin-2-one
N-[(3S,4R)-1-[2-(2-chloro-4-fluorophenyl)acetyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-ethoxy-4-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}phenol
1-[(4-methoxyphenyl)methyl]-4-(1-methyl-1H-pyrazole-5-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
1-(3,5-dimethylphenyl)-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-one
N-benzyl-3-{[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]oxy}benzamide
2-[3-(thiomorpholin-4-ylmethyl)phenoxy]acetamide
(3S,4R)-3-benzyl-1-(4-hydroxybenzoyl)-4-methylpiperidin-4-ol
(4aS,7aR)-1-[(2-fluoro-5-methoxyphenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-hydroxypropyl)-9-(1H-pyrazole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-N-pentyl-7-azaspiro[3.5]nonane-7-carboxamide
4,4,4-trifluoro-1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]butan-1-one
N,1-dimethyl-N-[3-(oxolan-2-yl)propyl]piperidin-4-amine