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1-(3-fluorobenzoyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-methanesulfonyl-N-methyl-4-(piperidin-3-yl)pyrimidin-2-amine
1-{3-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
4-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-phenylpiperazin-2-one
3-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-[4-(1H-pyrazol-5-yl)phenyl]urea
1-[(1-methylpiperidin-3-yl)methyl]-4-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperazine
4-(3-aminopyrrolidine-1-carbonyl)-N-(1,2-oxazol-3-ylmethyl)benzene-1-sulfonamide
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-2-methyl-4-phenylpyridine
2-cyclopentyl-9-(2-phenylacetyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
1-[(4-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}phenyl)methyl]-1H-1,2,3,4-tetrazole
1-methyl-4-(5-methyl-2H-1,2,3-triazole-4-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(1H-imidazol-2-yl)-N-[1-(1H-indol-2-yl)ethyl]-N-methylbenzamide
2-butyl-N-[(1-hydroxycyclohexyl)methyl]-1,3-benzoxazole-5-carboxamide
2-(4-fluorophenyl)-2-hydroxy-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}acetamide
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)pyridine-2-carboxamide
5-{[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-3-propyl-1,2-oxazole
(3S,4R)-1-(cyclobutylmethyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-(2-{1-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
4-(2-ethoxyphenyl)-3-(3,3,3-trifluoropropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-6-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-3-yl)pyrimidin-4-ol
4-benzyl-1-methyl-3-[1-(oxane-4-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
7-[ethoxy(phenyl)methyl]-4-(3-fluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(3,4-dimethoxyphenyl)methyl]-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
6-ethoxy-2-[4-(furan-3-ylmethyl)-1,4-diazepan-1-yl]-4-methylquinazoline
(1R,5S,6R)-3-cyclopentyl-N-(2-methoxyethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
(4-{[1-(2-methyl-5-propylpyrimidin-4-yl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
5-chloro-2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-1,3-benzodiazole
(4aS,8aR)-6-[2-(benzyloxy)acetyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(3-phenylpiperidin-1-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
(1S,5R)-3-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
8-chloro-2-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}quinoline
N-[(3,4-difluorophenyl)methyl]-3-(1-{[4-(2-hydroxyethoxy)phenyl]methyl}piperidin-3-yl)propanamide
9-(3-ethyl-1,2-oxazole-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-benzyl-9-propyl-2,9-diazaspiro[5.5]undecan-3-one
ethyl 4-{[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amino}piperidine-1-carboxylate
4-ethyl-3-{1-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-ethyl-3-[(1-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-1-(1-oxo-1,2-dihydroisoquinoline-4-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-[1-(methoxymethyl)cyclobutanecarbonyl]-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[(3-methoxyphenyl)methyl]-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}propanamide
6-methyl-N-[2-(oxan-2-yl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
4-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-cyclopentyl-1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carboxamide
ethyl 1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
[(5-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
5-(5-oxopyrrolidine-2-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide