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5-{[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
(3R,4R)-4-ethyl-1-{furo[3,2-c]pyridin-4-yl}piperidine-3,4-diol
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methyl-1,3-thiazol-2-yl)methyl]acetamide
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N,2,7,8-tetramethylquinoline-4-carboxamide
N-methyl-N-[2-(methylamino)ethyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(2-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{4-[2-(benzenesulfonyl)ethyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
N-[2-(2-fluorophenyl)ethyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-[1-(4-fluorophenyl)cyclopropanecarbonyl]-7-azaspiro[3.5]nonan-1-ol
5-{4-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
2-(4-cyclopentyl-1,4-diazepane-1-carbonyl)thiophene-3-sulfonamide
1-[(5-ethylpyridin-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(1H-pyrazol-1-yl)-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-4-carboxamide
N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)-2-(trifluoromethyl)benzamide
2-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(3-methoxyphenyl)piperazine
(1S,5R)-6-benzyl-3-{[4-(prop-2-en-1-yloxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-{6-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]pyridin-3-yl}ethan-1-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-fluoro-2-oxo-N-(propan-2-yl)-1,2-dihydroquinoline-4-carboxamide
[(4-cyclopropyl-5-{1-[(2-fluoro-4-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
1-cyclopropanecarbonyl-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}piperidine-4-carboxamide
6-(4-methoxyphenyl)-9-[2-(1,3-thiazol-4-yl)acetyl]-6,9-diazaspiro[4.5]decan-7-one
2-[3-(trifluoromethoxy)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(1R,3S)-3-(2-aminoethoxy)-7-(quinoline-3-carbonyl)-7-azaspiro[3.5]nonan-1-ol
1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(3-methylpyridin-4-yl)piperazine
2-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-6-ethoxyphenol
N-(2,5-dimethylphenyl)-3-(4H-1,2,4-triazol-4-yl)propanamide
(4aS,8aR)-1-(3-methoxypropyl)-6-(3-methylbut-2-enoyl)-decahydro-1,6-naphthyridin-2-one
3-[1-(2-oxo-2-phenylacetyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
2-(5-acetylthiophen-3-yl)-N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
ethyl 4-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperazine-1-carboxylate
N-[(2-fluorophenyl)methyl]-1-methyl-5-[4-(propan-2-yl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S)-3-benzyl-4-[(1-methyl-1H-imidazol-5-yl)methyl]piperazin-2-one
1-(3-{5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)-3-phenylprop-2-yn-1-one
3-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}benzonitrile
N-cycloheptyl-2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
N,1-diethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-[(5-chloro-2-propoxyphenyl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
2-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]pyridin-3-ol
4-({[4-(difluoromethoxy)phenyl]methyl}amino)-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
1-[7-(1-benzothiophen-3-yl)-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2,5-dimethoxyphenyl)ethan-1-one
8-(cyclohex-3-en-1-ylmethyl)-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,2-diphenylethyl)-3-(methanesulfonylmethyl)piperidine
5-{3-oxo-3-[4-(pyridin-3-yl)piperazin-1-yl]propyl}imidazolidine-2,4-dione