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2-methyl-N4-{2-[4-(3-methylbutoxy)phenyl]ethyl}pyrimidine-4,6-diamine
(3R,4S)-4-phenyl-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-amine
2-cyclopropyl-8-(2-{[(4-fluorophenyl)methyl](methyl)amino}acetyl)-2,8-diazaspiro[5.5]undecan-3-one
N-cyclobutyl-3-({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}sulfamoyl)benzamide
[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl][1-(ethylsulfanyl)propan-2-yl]amine
1-cyclobutyl-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(5-methylfuran-2-yl)benzamide
N-butyl-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
N-[1-(1H-imidazol-1-yl)butan-2-yl]-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
(3aR,5R,6S,7aS)-2-(5,8-dimethoxy-4-methylquinolin-2-yl)-octahydro-1H-isoindole-5,6-diol
7-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
(2S)-2-{[6-(2-aminoethyl)pyrimidin-4-yl]amino}-3-methylbutanamide
2-{4-[4-(2-methoxyphenyl)piperidin-1-yl]-5,6-dimethylthieno[2,3-d]pyrimidin-2-yl}ethan-1-amine
3-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridazine
3-{2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
(2R)-2-[(2-propyl-1,3-thiazol-4-yl)formamido]-3-(3,4,5-trifluorophenyl)propanoic acid
N-[2-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)ethyl]propanamide
9-[2-(1H-imidazol-1-yl)ethyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cycloheptyl-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-N,N-dimethylpiperidine-1-carboxamide
5-(5-ethylthiophen-2-yl)-2-propyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
9-ethyl-1-methyl-4-(1H-pyrrole-2-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N2,N2,5,6-tetramethyl-N4-[2-(pyridin-2-yl)ethyl]pyrimidine-2,4-diamine
3-(1-methyl-1H-pyrrol-2-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(2-methylphenyl)ethan-1-one
1-[5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carbonyl]-4-propyl-1,4-diazepane
8-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(2-fluorophenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine
(2S)-2-amino-1-[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-4-(methylsulfanyl)butan-1-one
3-{1-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
N-[2-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)quinolin-6-yl]acetamide
1-benzyl-4-oxo-N3-(prop-2-en-1-yl)-N5-[1-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-methyl-1,3-benzoxazole-6-carboxamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2,4-dimethyl-1,3-thiazole-5-carboxamide
(3S,9aR)-3-benzyl-2-methyl-8-[(4-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,7aR)-N-(3-fluorophenyl)-6,6-dioxo-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-4-methyl-1,3-oxazole-5-carboxamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-5-methoxy-1H-indole-2-carboxamide
(2S)-N-(2,3-dihydro-1H-inden-5-yl)-2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
(1S,6R)-9-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
8-methoxy-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(2-methylpropyl)-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
5-{1-[(6-chloro-2H-chromen-3-yl)methyl]pyrrolidin-2-yl}-N-methylthiophene-2-carboxamide
2-(2-chloro-5-fluorobenzoyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
6-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
1,3-dimethyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine