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3-(furan-2-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propan-1-one
2-({[4-(methylsulfanyl)phenyl]methyl}({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino)ethan-1-ol
1-{1-[5-(4-cyclohexylphenyl)-1,2,4-triazin-3-yl]piperidin-3-yl}ethan-1-one
(2R,3S,6R)-5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(4-{[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}phenyl)ethan-1-amine
(2E)-1-[(4aR,8aS)-6-(2-phenoxyacetyl)-decahydro-1,6-naphthyridin-1-yl]-3-(thiophen-2-yl)prop-2-en-1-one
5-(2,6-dimethoxyphenyl)-1-[3-(methylsulfanyl)propyl]-4-phenyl-1H-imidazole
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N,4,6-trimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(2S)-1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide
8-(5-methoxy-3-methyl-1H-indole-2-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(3aS,6aS)-5-(furan-3-carbonyl)-1-[(2E)-3-phenylprop-2-en-1-yl]-octahydropyrrolo[3,4-b]pyrrole
2-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
(2S,4S)-N-ethyl-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-(thiophene-3-amido)pyrrolidine-2-carboxamide
ethyl 2-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetate
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,4,6-trimethylpyrimidin-2-amine
1-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-[(4-hydroxypiperidin-1-yl)sulfonyl]-N-(pyrimidin-4-ylmethyl)benzamide
2-methyl-3-{[1-(pyridin-4-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-indole
(2-methoxyethyl)(oxolan-3-ylmethyl)[(2E)-3-phenylprop-2-en-1-yl]amine
2-(pyrrolidin-3-yl)-N-[2-(2,4,6-trimethylphenoxy)ethyl]acetamide
N,1,3-trimethyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(dimethylamino)-N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)acetamide
1-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}phenyl)-1H-pyrazole
2-acetyl-8-[5-(propan-2-yl)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3S,4R)-4-(3-fluorophenyl)-1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}pyrrolidine-3-carboxylic acid
4-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
5-(3-fluoro-2-methoxybenzoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
1-(cyclopropylmethyl)-5-[2-(2-fluorophenyl)acetyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,5R)-3-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{1-[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-yl]piperidin-3-yl}-3-methylbutan-1-one
[2-(2-methoxy-6-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}phenoxy)ethyl]dimethylamine
(2S,3S)-2-[(2-amino-5,6-dimethylpyrimidin-4-yl)amino]-3-methylpentanamide
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(furan-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(2-ethoxypyridin-3-yl)methyl]-2-ethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-{6-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
3-{3,4-dihydrospiro[1-benzopyran-2,1'-cyclohexane]-4-yl}-1-(2-hydroxypyridin-3-yl)urea
1-[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-[1-(furan-2-yl)ethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-(4-methyl-1H-pyrazol-1-yl)-N-(propan-2-yl)aniline
ethyl 4-[6-(2,3-dihydro-1-benzofuran-5-ylmethyl)-6-azaspiro[2.5]octane-1-carbonyl]piperazine-1-carboxylate
(4aS,8aR)-6-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(2-oxo-2-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethyl)pyrrolidin-2-one
(2S,4R)-N-(2-methoxyethyl)-1-(propan-2-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-{2-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-4-carboxamide
(1S,5R)-6-benzyl-3-(pent-2-yn-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3aR,6aR)-2-[3-(dimethylamino)benzoyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(3-methoxyphenyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-oxopiperazine-1-carboxamide
N3-(2-methoxyethyl)-N3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-1,3-dicarboxamide