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4-(6-methoxyquinolin-3-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-methyl-4-[1-(2-methylphenyl)piperidin-4-yl]piperazine-2-carboxylic acid
3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
4-(4-{[(3,5-dimethoxyphenyl)methyl]amino}piperidin-1-yl)-N-(1-phenylethyl)benzamide
3-{1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-4-yl}phenol
benzyl(cyclopropylmethyl){[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}amine
N-cyclopentyl-5-methyl-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-2-(propan-2-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-benzoxazole-5-carboxamide
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(3S,4S)-1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
6-(2-{[ethyl(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
1-(carbamoylmethyl)-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-3-carboxamide
2-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)formamido]ethyl}-4-methyl-1,3-thiazole-5-carboxylic acid
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-4-phenoxybutan-1-one
(1S,5R)-3-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
2-(3-chlorophenyl)-N-[4-(4-{[1-(thiophen-3-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]acetamide
1-ethyl-N-methyl-2-oxo-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1,2-dihydropyridine-4-carboxamide
1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidine-3-carboxamide
5-(morpholin-4-ylmethyl)-N-(2,2,2-trifluoroethyl)-1,2-oxazole-3-carboxamide
1-{1-oxa-8-azaspiro[4.6]undecan-8-yl}-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
3-{1-[(1-ethyl-1H-indol-3-yl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
2-(4-cyclohexyl-1,4-diazepan-1-yl)-2-(6-methoxypyridin-3-yl)acetic acid
4-benzyl-3-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-amino-6-(4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)-3,4-dihydropyrimidin-4-one
(2R,6R)-4-[(dimethyl-1,2-oxazol-4-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
9-(oxane-2-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-[(3-methoxyphenyl)methyl]-2-(2-methoxypyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decane
7-(oxan-4-yl)-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
[3-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-2,4,6-trimethylphenyl]methyl acetate
6-[3-(morpholin-4-ylmethyl)phenyl]quinazolin-4-amine
2-methyl-4-(3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)quinoline
N-[1-({[2-(1H-indol-1-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-(2-methoxyphenyl)propanamide
2-methoxy-5-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
N-(1-{7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
N-[(4-fluorophenyl)methyl]-N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3-methylbut-2-enamide
N-[(3R,4R)-1-(3-chloro-4-hydroxybenzoyl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
8-(pyrimidin-2-yl)-1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-1,8-diazaspiro[4.5]decane
methyl 9-(cyclopentyloxy)-7-oxo-3-[3-(1H-pyrazol-1-yl)propanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(6-hydroxy-1,4-oxazepan-4-yl)-2-(pyridin-4-ylsulfanyl)ethan-1-one
9-[(1R,9aR)-octahydro-1H-quinolizine-1-carbonyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}amine
4-chloro-2-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)phenol
3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1H-indazole
2-[(5-methylpyrazin-2-yl)methyl]-9-[(5-methylthiophen-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-4-{1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-imidazol-2-yl}piperidine
4-(8-methylquinolin-5-yl)pyridin-3-amine
N-[(2-chlorophenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine