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1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine
6-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyrimidin-4-amine
4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-(3,5-dimethylphenyl)piperazin-2-one
N-(pyridin-4-yl)quinoxaline-6-carboxamide
3-methyl-3-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-(2,4,6-trimethylpyridin-3-yl)urea
3-[1-(1-benzofuran-2-carbonyl)piperidin-3-yl]-N-[(3,4-difluorophenyl)methyl]propanamide
N'-(2-fluoro-5-methylphenyl)-N-(1-methanesulfonylpiperidin-4-yl)butanediamide
(3aR,6aS)-N-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
(3S,4S)-1-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-4-cyclopropylpyrrolidine-3-carboxylic acid
[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
4-(1-{1-[(2,4-dimethylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
3-(4-phenyl-1H-pyrazol-5-yl)-1-(1H-pyrazole-3-carbonyl)piperidine
1-(dimethylamino)-3-(4-{[methyl(thian-4-yl)amino]methyl}phenoxy)propan-2-ol
9-oxo-N-(propan-2-yl)-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
9-(2-acetylbenzoyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
4-[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-1-yl]phenol
6,8-dimethyl-2-({[4-(methylamino)butyl]amino}methyl)quinolin-4-ol
[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl](pyridin-2-yl)methanol
1-(2,3-dihydro-1H-inden-4-yl)-5-(1,3-thiazol-4-ylmethyl)-1H-1,2,4-triazole
4-{1-[(2-methoxyphenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3-methyl-1-propyl-1H-pyrazole
6-(3-methoxy-2-methylbenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(3R,4R)-1-(2H-1,3-benzodioxol-5-ylmethyl)-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-(thiophen-2-ylmethyl)piperidine
2-{[(3R,5S)-5-[4-(adamantan-2-yl)piperazine-1-carbonyl]-1-[(2,4-dimethoxy-3-methylphenyl)methyl]pyrrolidin-3-yl]sulfanyl}pyrimidine
1-{2-methyl-5-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
(3S,9aR)-3-benzyl-2-methyl-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
2-amino-4-(5-ethylfuran-2-yl)-6-(propan-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
methyl 3-{[(1R)-1-carbamoylethyl]carbamoyl}-5-(cyclobutylmethoxy)benzoate
4-benzyl-3-[1-(9H-purin-6-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,5R)-3-[(3-ethyl-1,2-oxazol-5-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
9-(3-chloropyridin-2-yl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-methyl-5-(3-methyl-3-phenylpiperidine-1-carbonyl)phenyl]imidazolidin-2-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidine
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]furan-2-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-[2-(pyridin-3-yloxy)phenyl]-1H-pyrazole-4-carboxamide
(1R,2R)-2-(4-{1-[2-(pyridin-2-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)cyclohexan-1-ol
1-{4-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}pyrrolidin-2-one
[(3R,5R)-1-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-(2-methylphenyl)pyrrolidin-3-ol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-6-methoxy-N,3-dimethyl-1-benzofuran-2-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(3-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
methyl 1-[(3R,5S)-5-[(1,3-dihydro-2-benzofuran-5-yl)carbamoyl]-1-[(2-methylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(4-methylphenoxy)ethyl]amine
3-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}pyridin-2-ol
(2S)-2-(methoxymethyl)-N-[2-(3-phenylpropoxy)phenyl]pyrrolidine-1-carboxamide
1-ethyl-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-6-oxopiperidine-3-carboxamide
5-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}-1,2-dihydropyridin-2-one
1-methyl-8-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid