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N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N,5,7-trimethyl-N-(oxolan-3-ylmethyl)pyrido[2,3-d]pyrimidin-4-amine
7-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1-oxa-7-azaspiro[3.5]nonane
(3aS,6aR)-5-(1,3-benzoxazol-2-yl)-3-cyclopentyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-methyl-5-[(2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-imidazol-1-yl)methyl]pyrrolidin-2-one
2-methoxy-N-{1-[3-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)phenyl]-1H-pyrazol-4-yl}acetamide
methyl 6-{[7-(2-methoxyacetyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}pyridine-2-carboxylate
2-{1-[(4-methylphenyl)methyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
2-(4-methyl-6-{[2-(pyrrolidin-1-yl)ethyl]amino}pyrimidin-2-yl)phenol
2-(3-hydroxypiperidin-1-yl)-1-[4-(3-methoxybenzoyl)piperazin-1-yl]ethan-1-one
2-methoxy-3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrazine
N-(2-hydroxy-2-phenylethyl)-4-{[2-(2-methoxyphenyl)ethyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
1-(2,3-dimethylphenyl)-4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
methyl 3-{[4-(1H-indole-2-carbonyl)-7-oxo-1,4-diazepan-1-yl]methyl}benzoate
1-[4-(5-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)propan-1-one
2-methyl-8-(4-methyl-1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3S,4R)-1-(2,3-dimethylquinoxaline-6-carbonyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
1-(furan-2-ylmethyl)-4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]pyridin-2-amine
(2-methoxyethyl)(methyl){[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
2-hydroxy-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
(4aS,8aR)-6-[(5-chlorothiophen-2-yl)methyl]-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
4-({5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)-N-methylbenzene-1-sulfonamide
(3S,4S)-1-[1-(furan-2-ylmethyl)piperidin-4-yl]-4-propylpyrrolidine-3-carboxylic acid
2-[2-benzyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]-N-ethylacetamide
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]piperidine-3-carboxamide
3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-1-(3-methylpiperidin-1-yl)propan-1-one
(4aS,7aR)-1-butyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(methoxymethyl)-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[5-(cyclohex-3-ene-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-cyclopropylpropanamide
3-[3-(morpholin-4-yl)-3-oxopropyl]-N-[2-(thiophen-2-yl)ethyl]piperidine-1-carboxamide
2-{4-[2-(9-methyl-9H-carbazol-3-yl)acetyl]morpholin-3-yl}acetic acid
11-{[2-(4-fluorophenyl)ethyl]amino}-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-methyl-3-(pyrrolidine-1-carbonyl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(1H-indazol-6-yl)-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperazin-2-one
2-(2-{[4-(2,4-difluorophenyl)piperazin-1-yl]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
(2S)-2-[(1-cyclohexylpiperidin-4-yl)formamido]-3-(pyridin-4-yl)propanoic acid
4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[(2,4-difluorophenyl)methyl]-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
5-(3-acetylphenoxymethyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
N-(3-cyclopentylpropyl)-5-(2,4-difluorophenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
(1S,9S)-11-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-benzyl-5-(1H-indol-2-ylmethyl)-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[3-(3-oxopiperazin-1-yl)propyl]-1-{4-[(trifluoromethyl)sulfanyl]phenyl}urea
4-methoxy-2-{[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
N-ethyl-N-[(2-fluorophenyl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide