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ethyl 5-({[1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)furan-2-carboxylate
2-{4-[4-(4-phenylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
N-[3-(4-methoxyphenyl)propyl]-1,3-dimethyl-1H-indole-2-carboxamide
4-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazine-1-carbonyl}pyridin-2-amine
N-methyl-N-(quinolin-2-ylmethyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-(3-methoxypropyl)-N-[(4-methylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-(2-{4-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
(3R,4S)-1-(4-methyl-1,3-thiazole-5-carbonyl)-4-propylpyrrolidin-3-amine
(3S,5S)-5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1-methylpyrrolidin-3-amine
1-{3-carboxy-5H,6H,7H-cyclopenta[b]pyridin-2-yl}-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
dimethyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})amine
4-methyl-6-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}pyrimidin-2-amine
1-(4-methoxyphenyl)-5-methyl-4-(3-phenoxypropanoyl)piperazin-2-one
methyl({[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl})[3-(oxolan-2-yl)propyl]amine
2-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2,3-dihydro-1H-isoindole
2-methoxy-N-[1-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
3-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-[(2-chlorophenyl)methyl]-4-hydroxy-N-(2-hydroxyethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(2H-1,3-benzodioxol-5-yl)-2-tert-butyl-1H-imidazole
3-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-N-(4-methoxyphenyl)-3-oxopropanamide
8-chloro-2-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)quinoline
2-(naphthalen-1-ylmethyl)-4-(thian-4-yl)morpholine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyridine-2-carboxamide
6-methyl-4-(4-methyl-1H-imidazol-5-yl)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-{5-[(4-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]urea
N-(2,2-diphenylethyl)-4-hydroxy-2-methylpyrimidine-5-carboxamide
1-(cyclopropylmethyl)-1',5',6',7'-tetrahydrospiro[azepane-4,4'-imidazo[4,5-c]pyridine]-7-one
3-oxo-N-propyl-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-ethyl-1,2-oxazole-5-carboxamide
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[3-(pyridin-3-yloxy)propyl]benzamide
ethyl 4-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
1-[(5-acetylthiophen-3-yl)methyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-(1,4-diazepane-1-sulfonyl)-N-(pyridin-3-yl)benzamide
(3S,4R)-1-(4-ethyl-5-methylthiophene-3-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-{1-[2-(3-methoxyphenyl)-1,3-benzoxazole-6-carbonyl]piperidin-3-yl}propan-1-one
1-(2-methoxyethyl)-8-[(3-methoxyphenyl)methyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(propan-2-yl)-1-(2-{1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-methylpiperidine-4-carbonitrile
[(3R,4S)-1-[(1-methyl-1H-indol-2-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-butyl-2-[(5,6-dimethylpyrimidin-4-yl)(methyl)amino]acetamide
1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
5-[4-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]-6-phenyl-2,3-dihydropyridazin-3-one
1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclopropan-1-amine
methyl 1-benzyl-5-[(furan-2-ylmethyl)amino]-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(2-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
8-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{[(4-methoxyphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5-methyl-5-phenylpiperidin-2-one
7-[(2-fluorophenyl)methyl]-2-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
3-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[3-(1H-1,2,4-triazol-1-yl)phenyl]urea