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1-[(4aR,8aR)-7-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-[(3,4-difluorophenyl)methyl]-3-[1-(3-phenoxypropanoyl)piperidin-3-yl]propanamide
N,N-dimethyl-9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-sulfonamide
3-(4-chloro-2-methylbenzoyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
2-methyl-N-[(5-methylpyrazin-2-yl)methyl]thieno[3,2-d]pyrimidin-4-amine
3-fluoro-5-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazine-1-carbonyl]benzonitrile
(3aR,6aR)-2-cyclopropanecarbonyl-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-chloro-N-cyclopentyl-4-{[1-(3-methyl-2-oxopentanoyl)piperidin-4-yl]oxy}benzamide
1-methyl-1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-5-yl]urea
(2S,4S)-4-amino-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,1-dimethylpyrrolidine-2-carboxamide
1-[5-(methylcarbamoyl)furan-2-yl]-3-phenyl-1H-pyrazole-4-carboxylic acid
5-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}quinoxaline
1-methyl-2-phenyl-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine
1-{[4-(hydroxymethyl)-4-[(4-methoxyphenyl)methyl]piperidin-1-yl]methyl}naphthalen-2-ol
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)propan-1-one
1-[3-(6-aminopyridin-2-yl)phenyl]propan-1-one
1-(benzylsulfamoyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-(1-butyl-4-methyl-1H-pyrazol-5-yl)acetamide
[3-(3-methylbut-2-en-1-yl)-1-(pyrrolidine-1-carbonyl)piperidin-3-yl]methanol
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(quinoline-2-carbonyl)pyrrolidin-3-yl]methanol
7-(1,3-benzothiazol-2-yl)-4-[(3-fluorophenyl)methyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1,3,7-trimethyl-2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
methyl 9-[2-(2-fluorophenyl)ethoxy]-7-oxo-3-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-1H-pyrazole-3-carboxylic acid
4-[(2-chloro-4,5-dimethoxyphenyl)methyl]-6-hydroxy-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-9-oxa-2-azaspiro[5.5]undecane
(1R,5S)-6-methyl-3-[(5-propylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(1-ethyl-1H-imidazol-2-yl)methyl]benzamide
8-(9H-purin-6-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
6-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}pyridine-2-carbonitrile
2-cyclopropanecarbonyl-8-(1-methyl-1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorothiophene-2-carboxamide
8-chloro-2-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
2-[2-(3-methylphenyl)pyrimidin-5-yl]-1H-1,3-benzodiazole-6-carboxylic acid
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(1-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
1,8-dimethyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2,5-dimethylphenyl)methyl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-(thiophen-3-ylmethyl)acetamide
{[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}(1H-imidazol-2-ylmethyl)amine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)-1-benzofuran-2-carboxamide
4-{3-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]propyl}-3,5-dimethyl-1H-pyrazole
(3aS,6aR)-5-(1,3-benzoxazol-2-yl)-3-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[1-(2,2-dimethylpropyl)-4-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
3-methyl-3-{4-[1-(pyrimidin-2-ylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}-1λ6-thiolane-1,1-dione
1-[2-(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)ethyl]pyrrolidin-2-one
(3aR,5R,6S,7aS)-2-[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]-octahydro-1H-isoindole-5,6-diol
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide