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1-(diethylamino)-3-(2-methoxy-5-{[methyl(oxan-4-yl)amino]methyl}phenoxy)propan-2-ol
(3aR,7aS)-2-(1-benzoxepine-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
3-methyl-5-{1-[3-(trifluoromethyl)phenoxy]ethyl}-1H-1,2,4-triazole
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-(propylsulfanyl)ethan-1-one
1-(5-chloropyridin-2-yl)-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperazine
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-[(oxan-4-yl)amino]pyridine-3-carboxamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3-(piperidin-1-yl)propan-1-one
2-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
1-[(1-{[1-(thian-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperidin-3-ol
2-{3-[2-(methoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}-4,7-dimethylquinazoline
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
(3aR,6aR)-2-methanesulfonyl-N-(2-phenoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[1-(pyridin-3-ylmethyl)azepan-4-yl]propanamide
N-[(2S,4R,6S)-2-[2-(carbamoylmethoxy)phenyl]-6-ethyloxan-4-yl]benzamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(4-chloro-1H-pyrazol-1-yl)propan-1-one
(3S)-1-(5-{[benzyl(methyl)amino]methyl}-1,2-oxazole-3-carbonyl)pyrrolidin-3-ol
N-(1-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
N-[(3-methoxyphenyl)methyl]-3-{1-[2-(3-methylphenyl)acetyl]piperidin-3-yl}propanamide
1-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-3-(thiophen-2-yl)propan-1-one
2-amino-4-(1-methyl-1H-pyrazol-4-yl)-6-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
2-[({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)amino]pyridine-3-carbonitrile
3-chloro-N-(2-methoxyethyl)-4-{[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]oxy}benzamide
N-benzyl-N-butyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
2-[benzyl(methyl)amino]-N-methyl-N-(pyrimidin-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
(3S,4R)-1-(2-methoxyethyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-[2-(pyrrolidine-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
3,6-dimethyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-benzofuran-2-carboxamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(1,3-benzothiazol-2-ylmethyl)propanamide
5-(morpholin-4-ylmethyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]furan-3-carboxamide
1-{5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}azepane
(4aR,7aS)-1-acetyl-4-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aR,8aR)-2-cyclobutanecarbonyl-7-(1H-imidazol-4-ylmethyl)-decahydro-2,7-naphthyridin-4a-ol
N-{[6-(2,3,4-trimethoxyphenyl)pyridin-3-yl]methyl}acetamide
3-[(dimethylamino)methyl]-1-[1-(pyridine-4-carbonyl)piperidine-4-carbonyl]pyrrolidin-3-ol
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
2-[(3,4-dimethyl-2-oxo-2H-chromen-7-yl)oxy]-N-(1H-imidazol-2-ylmethyl)-N-methylpropanamide
1-cyclopentyl-N-[2-(3-methoxyphenyl)ethyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4,6-dimethyl-3-[2-(4-methylpentyl)morpholine-4-carbonyl]-1,2-dihydropyridin-2-one
1-[4-({[4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)phenyl]pyrrolidin-2-one
2-phenyl-2-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-indene-1,3-dione
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N,N-bis(1,3-oxazol-4-ylmethyl)propanamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-benzyl-8-(3,3-dimethylcyclohexyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,5S)-5-(cyclopropylcarbamoyl)-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidine-3-carboxylic acid
(3S,4S)-1-[(2,4-difluorophenyl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
(2S,4R)-4-amino-N-methyl-1-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)pyrrolidine-2-carboxamide
N-(6-hydroxy-6-methylheptan-2-yl)-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(2,2,2-trifluoroethyl)butanamide