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3-[2-({5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)ethyl]-1,3-oxazolidin-2-one
(1R,7S)-3-(2-methoxyethyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-methyl-3-(4-{1-[2-(pyridin-2-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)-1λ6-thiolane-1,1-dione
N-[(3-{4-[(ethylcarbamoyl)amino]-3-methoxyphenyl}phenyl)methyl]propanamide
4-(pyridin-2-yl)-N-[1-(pyridin-3-yl)pentyl]pyrimidin-2-amine
ethyl 4-[(4-chlorophenyl)methyl]-1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidine-4-carboxylate
1-(2-methoxyethyl)-N-[2-(naphthalen-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-(3,3-diphenylpiperidin-1-yl)-2-methyl-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(3aS,6aS)-2-cyclopentyl-5-(2,5-difluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(1-benzylpiperidin-4-yl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-methyl-5-phenyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
(5-{1-[2-(piperidin-1-ylmethyl)phenyl]-1H-imidazol-2-yl}furan-2-yl)methanol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-6-methylpyridine-3-carboxamide
1-methanesulfonyl-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1,4-diazepane
(2R,3S,6R)-3-phenyl-5-(4-propylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[2-(morpholin-4-yl)pyridin-3-yl]-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl 4-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]butanoate
N-(1-{2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)methanesulfonamide
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-(1H-imidazol-1-yl)acetamide
2-{[(2,3-dimethyl-1H-indol-5-yl)methyl]amino}-N-(propan-2-yl)pyridine-4-carboxamide
(1-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
4-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-3-butyl-1-methylpiperazin-2-one
5-(3,3-dimethylbutyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
(2R,3R,6R)-5-(1H-imidazole-2-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{5-fluoro-7-[5-(propan-2-yl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(trifluoromethyl)phenyl]urea
N-{3-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-3-oxopropyl}-4-fluorobenzamide
1-[(2-phenyl-1H-imidazol-4-yl)methyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[1-(1H-1,2,4-triazol-5-yl)ethyl]amine
4-(2,4-dimethoxybenzoyl)-7-(pyridin-3-yl)-9-[2-(thiophen-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(1R)-1-(4-fluorophenyl)ethyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2,6,8-trimethyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}quinoline-4-carboxamide
2-[1-(2,2-dimethylpropyl)-4-(pyridin-3-ylmethyl)piperazin-2-yl]ethan-1-ol
1-cyclopentyl-N-ethyl-N-(2-methylprop-2-en-1-yl)-6-oxopiperidine-3-carboxamide
7-fluoro-N,2-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}quinoline-4-carboxamide
2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-methylacetamide
1-methyl-5-(1-phenylethyl)-3-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N,1,3-trimethyl-N-(1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-2-phenylethyl)-1H-pyrazole-5-carboxamide
4-chloro-N,N-diethyl-3-[2-(trimethyl-1H-pyrazol-1-yl)acetamido]benzamide
N-({7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
(7S,9aR)-N-benzyl-7-(cyclohexylmethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
5-[(2-fluorophenyl)methyl]-3-(3-methylbut-2-en-1-yl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-cyclopentyl-5-(morpholin-4-ylmethyl)-N-propyl-1,2-oxazole-3-carboxamide
5-({[(3-{2-[4-(2,5-dimethoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-dihydroquinolin-4-one
N-[5-(1H-pyrazol-4-yl)quinolin-8-yl]acetamide
3-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-3-methyl-1-[2-(methylsulfanyl)phenyl]urea
4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-3-(4-phenylphenyl)-1H-pyrazole
3-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridin-2-amine