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N-(oxolan-2-ylmethyl)-4-[({2-[(pyridin-3-yl)amino]ethyl}carbamoyl)amino]benzamide
N-(butan-2-yl)-2-methyl-N-(pyridin-2-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-chloro-N-{[1-(pyrimidin-2-ylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}pyridine-4-carboxamide
6-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carboxylic acid
{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}(ethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-ethyl-2-methoxy-N-[2-(4-methoxyphenoxy)ethyl]benzamide
N-butyl-2-[1-(5-cyclopropyl-1,3-oxazol-4-yl)-N-methylformamido]acetamide
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(1H-pyrazol-1-yl)butanamide
1-(carbamoylmethyl)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylpropanamide
1-ethyl-5-{2-[4-(propan-2-yl)morpholin-2-yl]acetyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)quinoline
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-4-(4-chlorophenyl)butan-1-one
(1S)-1-[1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
2-(1H-1,3-benzodiazol-1-yl)-N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]propanamide
N,5-dimethyl-4-{[(4-phenyloxan-4-yl)methyl]amino}-N-(1,3-thiazol-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
4-(3-fluorophenoxy)-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
(2E)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-phenylprop-2-enamide
methyl 3-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-2-yl)propanoate
1-[3-(3-cyclopropyl-1-propyl-1H-1,2,4-triazol-5-yl)propyl]azepane
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(dimethylamino)-N-methyl-2-(3-methylphenyl)acetamide
2-methoxy-5-{[3-(1H-pyrazol-5-yl)piperidin-1-yl]methyl}pyrimidine
8-(2,5-dimethylpyrimidin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-{2-[3-(4-chlorobenzoyl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
3-(3,4-dimethoxyphenyl)-N-[(3-methyloxetan-3-yl)methyl]propanamide
2-{4-[3-(methylsulfanyl)butyl]piperazin-1-yl}pyrazine
2-{[(2,4-difluoro-3-methoxyphenyl)methyl](thiophen-3-ylmethyl)amino}butan-1-ol
2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-phenyl-1,2-dihydrophthalazin-1-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(pyridin-2-ylmethyl)cyclopropanamine
4-[(1H-1,3-benzodiazol-2-ylmethyl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
2-methyl-7-[6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{3-[2-({[(4-fluorophenyl)methyl](methyl)amino}methyl)-4-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
3-(1-{[1-(3-methylbut-2-en-1-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-1-ol
N-(1-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
4-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
3-{5-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
5-butyl-1-(4-chlorophenyl)-4-(3-methyl-1,2-oxazole-5-carbonyl)piperazin-2-one
N-[(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine-2-carboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)-3-[(thiophen-2-ylmethyl)amino]benzamide
4,6-dimethyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N3-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-N1-(pyridin-3-yl)propane-1,3-diamine
1-{1-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}piperidin-3-ol
2-{4-[6-ethyl-4-(4-methylpiperidine-1-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
3-(2-methoxyethyl)-1-(4-methylquinolin-2-yl)piperidine-3-carboxylic acid
(2S,4S)-4-[2-(1H-1,3-benzodiazol-2-yl)acetamido]-1-methylpyrrolidine-2-carboxylic acid
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)propanamide
1-cyclopentyl-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-diazepane
4-(6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carbonyl)morpholine