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5-tert-butyl-4-[(1-oxo-1,2-dihydrophthalazin-2-yl)methyl]furan-2-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}propanamide
9-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
2-{1-cyclohexyl-4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
6-(4-methylpiperazin-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
5-{1-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}-2-methoxybenzoic acid
6-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
methyl 4-[(3-{[(2,5-dimethylfuran-3-yl)formamido]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)methyl]benzoate
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]propanamide
(3aR,6aR)-N-[2-(tert-butylsulfanyl)ethyl]-2-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)-2-[3-(2-methylphenoxy)azetidin-1-yl]pyrimidine
6-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
7-(1,3-benzothiazol-2-yl)-4-(3-chloro-4-fluorobenzenesulfonyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-methyl-6-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1H,2H-pyrazolo[1,5-a]pyrimidin-2-one
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
3-methyl-8-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
6-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
2-(cyclohexylmethyl)-4-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}morpholine
1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
5-{5-[4-(1H-pyrazol-3-yl)phenyl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
4-(1-butyl-1H-imidazol-2-yl)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidine
2-{[7-(2-propylpyridine-4-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
7-({ethyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2-methoxypyridine-3-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-phenylacetamide
1-{4-[4-(thian-4-yl)piperazine-1-carbonyl]phenyl}pyrrolidin-2-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-(piperidin-1-ylmethyl)piperidin-2-one
2-[2-(3-fluorophenyl)-2-oxoethyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
{7-fluoro-5-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-(2-{2-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}ethyl)-1,3-oxazinan-2-one
(1R,5S,8R)-3-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-azabicyclo[3.2.1]octan-8-ol
N-benzyl-5-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)pyrimidin-2-amine
N-methyl-6-oxo-1-(2-phenylethyl)-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-3-carboxamide
8-(1,3-benzothiazol-2-ylmethyl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[2-(2,6-difluorophenyl)ethyl]-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-4-(quinolin-7-ylmethyl)-1,4-diazepan-2-one
1-[1'-(6-methoxypyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
7-(3-phenylpropyl)-2-[2-(1H-pyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
N,4-dimethyl-1-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidine-4-carboxamide
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,6-dichlorobenzamide
methyl 7-oxo-3-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(aminomethyl)-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
1-(1-cyclohexanecarbonylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-(2,3-dihydro-1H-inden-5-yloxy)-2-methyl-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}propan-1-one
2-(2-{[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propanoic acid
N-ethyl-N-methyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
(2E)-1-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-3-(pyridin-4-yl)prop-2-en-1-one