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4-[(3-chloropyridin-4-yl)methyl]-2-(2-methoxyethyl)morpholine
4-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-1,2-dihydrophthalazin-1-one
2-(2-chlorophenyl)-2-[(2-oxo-1,2-dihydroquinolin-4-yl)formamido]acetic acid
N-(2-methoxyethyl)-N-methyl-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
6-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
5-{1-[(5-cyclohexylthiophen-2-yl)methyl]pyrrolidin-2-yl}-3-methyl-1H-1,2,4-triazole
N2-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(pyridin-3-yl)ethane-1,2-diamine
(1S,6R)-9-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)[3-(methylsulfanyl)propyl]amine
(2,3-dihydro-1-benzofuran-2-ylmethyl)({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
(1,4-dioxan-2-ylmethyl)(methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
N-(3-methoxypropyl)-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[(3-methylphenyl)methyl]-4-{[3-(pyridin-2-yl)phenyl]methyl}piperazine
2-(3-methylbut-2-en-1-yl)-8-(4-oxo-4-phenylbutyl)-2,8-diazaspiro[4.5]decan-3-one
[(3R,5R)-1-[2-(methylsulfanyl)pyridine-3-carbonyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
1,3-dimethyl-8-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1R,9S)-5-amino-3-(6-ethoxypyridin-3-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
(1R,5S,6R)-3-{[4-(cyclopentyloxy)phenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
N-(2-methoxyethyl)-4-methyl-N-[(3-methylthiophen-2-yl)methyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-butyl-N-methylpiperidine-3-carboxamide
3-amino-N-[1-(thiophen-2-yl)butyl]benzamide
N-[(3S,4R)-1-[2-(2,4-dimethoxyphenyl)acetyl]-4-propylpyrrolidin-3-yl]acetamide
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}[(2-methylpyrimidin-5-yl)methyl]amine
2-cyclopropyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1,3-benzoxazole-6-carboxamide
1-[2-(3-fluorophenyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N4,N4-diethyl-N6-[(4-methanesulfonylmorpholin-2-yl)methyl]pyrimidine-2,4,6-triamine
5-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]pyrazin-2-ol
1-[2-oxo-2-(3-propylmorpholin-4-yl)ethyl]imidazolidine-2,4-dione
1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-3-phenylpyrrolidin-3-ol
(1S,3R)-3-amino-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}cyclopentane-1-carboxamide
2-[(2,3-dihydro-1H-inden-5-ylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-butyl-4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N3-[(5-chlorothiophen-2-yl)methyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-(furan-3-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
3-{[(1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
5-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidine-1-carbonyl}-N-(propan-2-yl)pyrimidin-2-amine
1-(4-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-[5-(methoxymethyl)furan-2-carbonyl]-3-(4-phenylbenzoyl)piperidine
3-[(1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperidin-4-yl)oxy]pyridine
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
(3R,4S)-4-(4-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-1,4-diazepan-1-yl)oxolan-3-ol
1-(dimethylamino)-2-[4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-2-ol
2-cyclopentyl-8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-({6-[4-(1H-pyrazol-1-yl)phenyl]pyridin-3-yl}methyl)morpholine
N-cyclooctyl-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
methyl 3-[4-(2-chloro-4-fluorobenzoyl)-6-[(3-methoxyphenyl)methoxy]-2-oxo-1,4-diazepan-1-yl]propanoate
N-cyclopropyl-2-(dimethylamino)-2-(3-methylphenyl)-N-(1,3-thiazol-5-ylmethyl)acetamide