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6-methyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
6-[(2S)-2-carbamoylpyrrolidin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}(methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
1-[2-(3-methoxypropyl)piperidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(3-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-chloro-N-[2-(dimethylamino)ethyl]-N-(2-hydroxyethyl)-5-(1H-pyrazol-1-yl)benzamide
(3aR,6aR)-2-(dimethyl-1,3-thiazole-5-carbonyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({7-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
2-(1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
2-(4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-cyclohexylpiperazin-2-yl)ethan-1-ol
(1R,6S)-9-methyl-3-(pyridine-3-sulfonyl)-3,9-diazabicyclo[4.2.1]nonane
1-(2-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
3-(5-methyl-1H-pyrazol-1-yl)-1-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
1-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
4-[(2-chloro-6-fluorophenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(2S)-2-{4-[5-(2-cyanophenyl)furan-2-yl]-1H-1,2,3-triazol-1-yl}-3-methylbutanamide
5-methyl-1-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-5-phenylpiperidin-2-one
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl][(2,3-difluoro-6-methoxyphenyl)methyl]methylamine
1-ethyl-8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[4-(1H-1,3-benzodiazol-1-yl)phenyl]-1-(1,4-oxazepan-6-ylmethyl)urea
[2-(1H-imidazol-1-yl)ethyl](methyl){[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
N-[4-(morpholin-4-ylmethyl)phenyl]-3-phenylpiperazine-1-carboxamide
3-[4-(pyridin-4-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroisoquinolin-1-one
3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
(3R,5S)-N-[3-(dimethylamino)propyl]-5-(3-fluorophenoxymethyl)-1-(2-phenylethyl)piperidine-3-carboxamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(3-phenylpiperidin-1-yl)acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(phenylamino)pyrimidine-5-carboxamide
N-(furan-2-ylmethyl)-N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetamide
1-{2-[2-(pyridin-2-yl)ethyl]phenyl}-3-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
(1S,6R)-3-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
[2-(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)phenyl]methanol
4-({1-[(2R)-2-aminopropanoyl]piperidin-4-yl}oxy)-3-chloro-N-(2-methoxyethyl)benzamide
4-[(2-amino-6-methylpyrimidin-4-yl)amino]-1-[(2-chlorophenyl)methyl]pyrrolidin-2-one
5-(2,6-dimethylphenoxymethyl)-N,N-bis(prop-2-en-1-yl)-1,2-oxazole-3-carboxamide
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-(2-methoxyethoxy)ethan-1-one
1-{[2-(3-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}azetidin-3-ol
7-methoxy-4-(2-methylpyrrolidine-1-carbonyl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline
2-(2-cyclopropylpyrimidin-5-yl)-N-ethyl-7-methyl-N-(propan-2-yl)quinoline-4-carboxamide
2-(3-chlorophenyl)-N-(2,3-dihydro-1H-inden-2-yl)-2-hydroxy-N-methylacetamide
2-(4-acetyl-1,4-diazepan-1-yl)-2-(2-butoxy-4-fluorophenyl)acetic acid
4-(furan-3-ylmethyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
(1H-1,3-benzodiazol-2-ylmethyl)(ethyl)({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amine
2-({6-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1-methyl-1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N-ethylpyrimidin-4-amine
1-benzyl-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]piperidin-4-amine
4-{4-oxo-7-[2-(pyrimidin-2-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
3-cyclopentyl-5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2,3-dimethyl-7-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one