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5-{[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
1-cyclopropanecarbonyl-4-[4-(3-methoxypiperidine-1-carbonyl)phenoxy]piperidine
(1S,5R)-3-benzoyl-6-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
1-(3-methylpyridin-4-yl)-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
1-(3-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
2-(2-methoxyethyl)-4-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}morpholine
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-[3-(methoxymethyl)pyrrolidin-1-yl]pyridine
5-(pyridin-4-yl)-N-(2,2,2-trifluoroethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[1-(5-ethyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
N6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-9H-purine-2,6-diamine
4-[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carbonyl]-1,4-diazepan-2-one
N-cyclopropyl-N-({4-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(1-cycloheptylpiperidin-3-yl)-4-(4-methoxyphenyl)piperazine
N-cyclopropyl-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N,N-diethyl-1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxamide
1-[4-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)thiophen-2-yl]ethan-1-one
4-{[4-(difluoromethoxy)phenyl]methyl}-6-methoxy-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2,5-dimethyl-3-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
N-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
N-{[5-fluoro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
N-[(2R,3R)-1'-[(2-hydroxy-5-methoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
5-cyclohexaneamido-N-[(3-fluorophenyl)methyl]-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-methoxypropan-1-one
3-amino-1-{[3-(morpholin-4-ylmethyl)phenyl]methyl}pyrrolidine-3-carboxylic acid
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(9H-purin-6-yl)piperidin-3-amine
1-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
5-(2-chlorophenyl)-N-[1-(1,3-thiazol-5-yl)propan-2-yl]furan-2-carboxamide
N-{[1-(3-methylpyridin-2-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}benzamide
ethyl 6-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylate
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-[({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)amino)methyl]piperidin-2-one
4-{5-methyl-2-oxo-4-[3-(piperidin-1-yl)propanoyl]piperazin-1-yl}benzonitrile
4-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl}benzene-1-sulfonamide
N-[(3-chloro-4-fluorophenyl)methyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-(4-{3-[(2-methoxyethyl)carbamoyl]piperidin-1-yl}piperidin-1-yl)pyridine-3-carboxamide
(3E)-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-3-en-1-one
2-{1-cyclopentyl-4-[3-(hydroxymethyl)-8-methylquinolin-2-yl]piperazin-2-yl}ethan-1-ol
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
N-cyclopentyl-2-({[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)propanamide
5-methyl-4-oxo-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
1-(dimethylamino)-3-(4-methoxy-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenoxy)propan-2-ol
(5S,9aS,9bS)-2-methyl-5-[2-(trifluoromethyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[3-(1H-imidazol-4-yl)-2-(1H-pyrrol-1-yl)propanoyl]-1-phenylpiperazin-2-one
2-(2-aminoethyl)-N-cyclopropyl-N-(1,3-thiazol-2-ylmethyl)quinazolin-4-amine
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(2,5-dimethoxyphenyl)pyrrolidine
{[2-(2-methoxyphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}(thiophen-2-ylmethyl)amine
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)acetamide
2-({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}amino)butan-1-ol
N-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methanesulfonamide
5-[2-(methylsulfanyl)phenoxymethyl]-N-(3-phenylpropyl)-1,2-oxazole-3-carboxamide
3-(2-methoxyethyl)-5-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazole