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1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
N-(3-methoxyphenyl)-3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-N-(2,2,2-trifluoroethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(propan-2-yl)-1-(2-{1-[3-(pyridin-3-yl)propanoyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
3-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
ethyl 1-[2-(methylsulfanyl)acetyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
1-ethyl-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]urea
3-{1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}benzoic acid
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
1-{4-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
6-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}imidazo[1,2-a]pyridine-2-carboxamide
(3R,5S)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
2-(1,1-dioxo-1λ6-thian-4-yl)-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]acetamide
(1S,5R)-6-(1-methyl-1H-pyrazole-3-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[4-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]phenol
methyl 3-(2-methoxyacetamido)-5-[(3-methylbut-2-en-1-yl)amino]-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(1,3-benzothiazol-5-yl)-4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}propanamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
(3S,4R)-1-[2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N3-tert-butyl-1-(3-methylbutyl)-4-oxo-N5-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(pyrrolidin-1-yl)-3-[1-(thiolan-3-yl)piperidin-4-yl]propan-1-one
N-cyclobutyl-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
7-(2-methylphenyl)-4-(pyrimidin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{4-[4-(2-amino-6-methylpyrimidin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
2-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
(5-{[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}furan-2-yl)methanol
5-{1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]pyrrolidin-2-yl}-N-ethylthiophene-2-carboxamide
4-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-ethyl-1H-pyrazole
6-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
2-cyclopentyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
methyl (2S)-3-carbamoyl-2-{2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}propanoate
ethyl 2-(1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-N-methylformamido)acetate
6-{[benzyl(methyl)amino]methyl}-2-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
N-[3-(furan-2-yl)phenyl]-1-(thiophene-3-carbonyl)piperidine-4-carboxamide
N-{1-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-1H-pyrazol-4-yl}-2-phenoxyacetamide
(4aS,8aR)-6-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(4-methoxyphenyl)methyl]-7-methyl-N-(oxolan-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide
ethyl 4-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-2-(pyridin-2-yl)acetamide
2-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methoxy}benzamide
3-(5-methylthiophen-2-yl)-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-pyrazole
4-{4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxybenzoyl}-1,4-diazepane-1-carbaldehyde
N-[4-(furan-2-yl)phenyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine-3-carboxamide
7-(5-chloropyridin-2-yl)-4-[1-(methoxymethyl)cyclopropanecarbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]propanoic acid
N-ethyl-2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N-methylpyrimidin-4-amine